PDB ID: 4EBV
Hetero Atom Contents
color scheme of protein:
hetatm:
x
information
centroid:
interaction residue:
chain:
Structure summary
Code : | 4EBV PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | Structure of Focal Adhesion Kinase catalytic domain in complex with novel allosteric inhibitor | ||||||||||||
Release Data : | 2012-08-22 | ||||||||||||
Compound : |
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Source : |
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Authors : | Skene, R.J., Hosfield, D.J. | ||||||||||||
Keywords : | Kinase Domain, Allosteric inhibitor, TRANSFERASE-TRANSFERASE INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.67 Å ) | ||||||||||||
Citation : |
Discovery and characterization of novel allosteric FAK inhibitors.
Iwatani, M.,Iwata, H.,Okabe, A.
et al.
PubMed: 22819505 |
Reaction
Chain : | A |
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UniProt : | Q05397 (FAK1_HUMAN) |
Reaction : | Reaction=ATP + L-tyrosyl-[protein] = ADP + H(+) + O-phospho-L-tyrosyl- [protein]; Xref=Rhea:RHEA:10596, Rhea:RHEA-COMP:10136, Rhea:RHEA- COMP:10137, ChEBI:CHEBI:15378, ChEBI:CHEBI:30616, ChEBI:CHEBI:46858, ChEBI:CHEBI:82620, ChEBI:CHEBI:456216; EC=2.7.10.2; Evidence={ECO:0000255|PROSITE-ProRule:PRU10028, ECO:0000269|PubMed:10655584, ECO:0000269|PubMed:11331870, ECO:0000269|PubMed:18339875}; |