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Ligands
Code Name Style Show Link
CPR 6-chloropurine riboside, 5'-monophosphate
SAE Selenazole-4-carboxyamide-adenine dinucleotide
Non-standard Residues
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Glycosylation
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Code : 1B3O   PDBj   RCSB PDB   PDBe
Header : DEHYDROGENASE
Title : TERNARY COMPLEX OF HUMAN TYPE-II INOSINE MONOPHOSPHATE DEHYDROGENASE WITH 6-CL-IMP AND SELENAZOLE ADENINE DINUCLEOTIDE
Release Data : 1999-04-12
Compound :
mol_id molecule chains synonym
1 PROTEIN (INOSINE MONOPHOSPHATE DEHYDROGENASE 2) A,B IMPD, IMPDH
ec: 1.1.1.205
Source :
mol_id organism_scientific organism_common expression_system
1 Homo sapiens  (taxid:9606) Human Escherichia coli  (taxid:562)
variant: TYPE II ISOZYME
Authors : Colby, T.D., Vanderveen, K., Strickler, M.D., Goldstein, B.M.
Keywords : DEHYDROGENASE, IMPD, IMPDH, GUANINE NUCLEOTIDE SYNTHESIS
Exp. method : X-RAY DIFFRACTION ( 2.90 Å )
Citation :

Crystal structure of human type II inosine monophosphate dehydrogenase: implications for ligand binding and drug design.

Colby, T.D.,Vanderveen, K.,Strickler, M.D.  et al.
(1999)  Proc.Natl.Acad.Sci.USA  96 : 3531 - 3536

PubMed: 10097070
DOI: 10.1073/pnas.96.7.3531

Chain : A, B
UniProt : P12268 (IMDH2_HUMAN)
Reaction: EC: Evidence:
Physiological Direction:
H2O + IMP + NAD(+) = H(+) + NADH + XMP 1.1.1.205 PubMed:7763314, PubMed:7903306
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