PDB ID: 3WIG
Hetero Atom Contents
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Code | Name | Style | Show | Link | |
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ANP | Phosphoaminophosphonic acid-adenylate ester | PoSSuM | |||
MG | Magnesium ion | PoSSuM | |||
CHU | N-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-N'-methylsulfuric diamide | PoSSuM | |||
PG4 | Tetraethylene glycol | PoSSuM | |||
CL | Chloride ion | PoSSuM |
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Download interaction data: 3WIG
Structure summary
Code : | 3WIG PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | Human MEK1 kinase in complex with CH5126766 and MgAMP-PNP | ||||||||||||
Release Data : | 2014-06-04 | ||||||||||||
Compound : |
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Source : |
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Authors : | Lukacs, C.M., Janson, C., Schuck, V. | ||||||||||||
Keywords : | kinase, kinase inhibitor, allosteric, TRANSFERASE-TRANSFERASE INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.7000 Å ) | ||||||||||||
Citation : |
Disruption of CRAF-Mediated MEK Activation Is Required for Effective MEK Inhibition in KRAS Mutant Tumors
Lito, P.,Saborowski, A.,Yue, J.
et al.
PubMed: 24746704 |
Reaction
Chain : | A | ||||||||||||||||
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UniProt : | Q02750 (MP2K1_HUMAN) | ||||||||||||||||
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