ID 5VK1A STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 26 49 VAL A 13 12 PRO B Protein S 2 FT #SUB 26 49 VAL A 14 13 NH2 B Protein S 1 FT #SUB 27 50 LYS A 13 12 PRO B Protein A 2 FT #SUB 27 50 LYS A 14 13 NH2 B Protein B 2 FT #SUB 30 53 MET A 8 7 TRP B Protein A 4 FT #SUB 30 53 MET A 12 11 SER B Protein S 1 FT #SUB 30 53 MET A 13 12 PRO B Protein S 1 FT #SUB 34 57 GLY A 4 3 PHE B Protein B 1 FT #SUB 34 57 GLY A 8 7 TRP B Protein B 8 FT #SUB 37 60 ILE A 4 3 PHE B Protein S 4 FT #SUB 43 66 TYR A 4 3 PHE B Protein S 2 FT #SUB 48 71 GLN A 3 2 SER B Protein S 3 FT #SUB 48 71 GLN A 4 3 PHE B Protein A 11 FT #SUB 49 72 HIS A 7 6 TYR B Protein A 4 FT #SUB 69 92 VAL A 4 3 PHE B Protein S 1 FT #SUB 69 92 VAL A 7 6 TYR B Protein S 1 FT #SUB 69 92 VAL A 11 10 LEU B Protein B 1 FT #SUB 72 95 PRO A 11 10 LEU B Protein S 1 FT #SUB 75 98 LEU A 8 7 TRP B Protein S 1 FT #SUB 71 94 ASP A 27 50 LYS C Protein S 6 FT #SUB 73 96 SER A 25 48 THR C Protein S 4 FT #SUB 76 99 TYR A 2 25 ASN C Protein S 12 FT #SUB 70 93 LYS A 13 12 PRO D Protein S 7 FT #SUB 70 93 LYS A 14 13 NH2 D Protein S 2 FT #SUB 7 30 LYS A 39 62 VAL G Protein S 5 FT #SUB 60 83 GLU A 45 68 ALA G Protein S 1 FT #SUB 81 104 LYS A 41 64 GLN G Protein B 1 FT #SUB 82 105 ASN A 41 64 GLN G Protein S 3 FT #SUB 2 25 ASN A 26 49 VAL I Protein S 2 FT #SUB 2 25 ASN A 80 103 ARG I Protein B 2 FT #SUB 26 49 VAL A 10 9 LEU J Protein S 1 FT #SUB 26 49 VAL A 11 10 LEU J Protein S 4 FT #SUB 26 49 VAL A 13 12 PRO J Protein S 1 FT #SUB 30 53 MET A 10 9 LEU J Protein S 2 FT #SUB 76 99 TYR A 9 8 CYS J Protein S 2 FT #SUB 76 99 TYR A 13 12 PRO J Protein S 3 FT #SUB 76 99 TYR A 14 13 NH2 J Protein S 3 FT #SUB 79 102 LEU A 13 12 PRO J Protein S 1 FT #SUB 80 103 ARG A 14 13 NH2 J Protein A 3 FT DISORDER 1 1 FT DISORDER 85 85 CC SEQUENCE 83 AA (ATOM); CC NQVRPKLPLL KILHAAGAQG EMFTVKEVMH YLGQYIMVKQ LYDAAAQHMV YCGGDLLGEL CC LGRQSFSVKD PSPLYDMLRK NLV CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM -NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************* CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV- CC ********************************** SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1B STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 3 2 SER B 48 71 GLN A Protein A 3 FT #SUB 4 3 PHE B 34 57 GLY A Protein S 1 FT #SUB 4 3 PHE B 37 60 ILE A Protein S 4 FT #SUB 4 3 PHE B 43 66 TYR A Protein S 2 FT #SUB 4 3 PHE B 48 71 GLN A Protein A 11 FT #SUB 4 3 PHE B 69 92 VAL A Protein S 1 FT #SUB 7 6 TYR B 49 72 HIS A Protein S 4 FT #SUB 7 6 TYR B 69 92 VAL A Protein S 1 FT #SUB 8 7 TRP B 30 53 MET A Protein S 4 FT #SUB 8 7 TRP B 34 57 GLY A Protein S 8 FT #SUB 8 7 TRP B 75 98 LEU A Protein S 1 FT #SUB 11 10 LEU B 69 92 VAL A Protein S 1 FT #SUB 11 10 LEU B 72 95 PRO A Protein S 1 FT #SUB 12 11 SER B 30 53 MET A Protein B 1 FT #SUB 13 12 PRO B 26 49 VAL A Protein B 2 FT #SUB 13 12 PRO B 27 50 LYS A Protein S 2 FT #SUB 13 12 PRO B 30 53 MET A Protein B 1 FT #SUB 14 13 NH2 B 26 49 VAL A Protein B 1 FT #SUB 14 13 NH2 B 27 50 LYS A Protein B 2 FT #SUB 9 8 CYS B 70 93 LYS I Protein B 2 FT #SUB 10 9 LEU B 70 93 LYS I Protein B 2 FT #SUB 12 11 SER B 69 92 VAL I Protein S 1 FT #SUB 13 12 PRO B 69 92 VAL I Protein S 1 FT #SUB 13 12 PRO B 70 93 LYS I Protein S 5 FT #SUB 13 12 PRO B 72 95 PRO I Protein S 1 FT #SUB 10 9 LEU B 7 6 TYR J Protein B 2 FT #SUB 12 11 SER B 7 6 TYR J Protein S 6 FT #SUB 12 11 SER B 10 9 LEU J Protein A 3 FT #SUB 12 11 SER B 11 10 LEU J Protein S 2 FT #SUB 13 12 PRO B 10 9 LEU J Protein B 3 FT #SUB 13 12 PRO B 11 10 LEU J Protein B 2 FT #SUB 14 13 NH2 B 11 10 LEU J Protein B 2 CC SEQUENCE 14 AA (ATOM); CC XTSFXEYWCL LSPX CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLLSPX CC ************** SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX // ID 5VK1C STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 2 25 ASN C 76 99 TYR A Protein A 12 FT #SUB 25 48 THR C 73 96 SER A Protein S 4 FT #SUB 27 50 LYS C 71 94 ASP A Protein S 6 FT #SUB 27 50 LYS C 13 12 PRO D Protein S 3 FT #SUB 30 53 MET C 8 7 TRP D Protein B 4 FT #SUB 30 53 MET C 11 10 LEU D Protein S 1 FT #SUB 30 53 MET C 12 11 SER D Protein S 3 FT #SUB 33 56 LEU C 8 7 TRP D Protein S 1 FT #SUB 34 57 GLY C 4 3 PHE D Protein B 1 FT #SUB 34 57 GLY C 8 7 TRP D Protein B 7 FT #SUB 37 60 ILE C 4 3 PHE D Protein S 6 FT #SUB 38 61 MET C 4 3 PHE D Protein S 1 FT #SUB 38 61 MET C 5 4 9E7 D Protein S 2 FT #SUB 43 66 TYR C 4 3 PHE D Protein S 2 FT #SUB 48 71 GLN C 2 1 THR D Protein S 2 FT #SUB 48 71 GLN C 3 2 SER D Protein S 2 FT #SUB 48 71 GLN C 4 3 PHE D Protein A 5 FT #SUB 49 72 HIS C 7 6 TYR D Protein A 11 FT #SUB 69 92 VAL C 4 3 PHE D Protein S 1 FT #SUB 69 92 VAL C 7 6 TYR D Protein S 3 FT #SUB 69 92 VAL C 8 7 TRP D Protein S 1 FT #SUB 69 92 VAL C 11 10 LEU D Protein A 2 FT #SUB 72 95 PRO C 11 10 LEU D Protein S 1 FT #SUB 76 99 TYR C 11 10 LEU D Protein S 1 FT #SUB 70 93 LYS C 20 43 GLN E Protein S 4 FT #SUB 70 93 LYS C 21 44 GLY E Protein A 2 FT #SUB 70 93 LYS C 23 46 MET E Protein S 3 FT #SUB 70 93 LYS C 24 47 PHE E Protein S 7 FT #SUB 70 93 LYS C 28 51 GLU E Protein S 5 FT #SUB 2 25 ASN C 5 4 9E7 J Protein S 2 FT #SUB 50 73 MET C 15 38 HIS K Protein S 2 FT #SUB 52 75 TYR C 8 31 LEU K Protein S 2 FT #SUB 52 75 TYR C 12 35 LYS K Protein S 1 FT #SUB 52 75 TYR C 15 38 HIS K Protein S 4 FT #SUB 54 77 GLY C 8 31 LEU K Protein B 2 FT #SUB 55 78 GLY C 8 31 LEU K Protein B 1 FT #SUB 64 87 ARG C 22 45 GLU K Protein A 16 FT #SUB 65 88 GLN C 6 29 PRO K Protein S 3 FT #SUB 65 88 GLN C 7 30 LYS K Protein S 2 FT #SUB 65 88 GLN C 8 31 LEU K Protein A 4 FT #SUB 65 88 GLN C 22 45 GLU K Protein B 1 FT #SUB 66 89 SER C 11 34 LEU K Protein S 2 FT #SUB 66 89 SER C 15 38 HIS K Protein S 1 FT #SUB 66 89 SER C 22 45 GLU K Protein B 3 FT #SUB 64 87 ARG C 71 94 ASP M Protein S 1 FT #SUB 64 87 ARG C 73 96 SER M Protein S 1 FT #SUB 71 94 ASP C 64 87 ARG M Protein S 2 FT #SUB 71 94 ASP C 71 94 ASP M Protein S 3 FT #SUB 71 94 ASP C 74 97 PRO M Protein S 1 FT #SUB 73 96 SER C 73 96 SER M Protein S 3 FT #SUB 73 96 SER C 74 97 PRO M Protein S 2 FT #SUB 74 97 PRO C 73 96 SER M Protein S 1 FT #SUB 80 103 ARG C 80 103 ARG M Protein S 11 FT DISORDER 1 1 FT DISORDER 84 85 CC SEQUENCE 82 AA (ATOM); CC NQVRPKLPLL KILHAAGAQG EMFTVKEVMH YLGQYIMVKQ LYDAAAQHMV YCGGDLLGEL CC LGRQSFSVKD PSPLYDMLRK NL CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM -NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************* CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNL-- CC ********************************* SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1D STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 13 12 PRO D 70 93 LYS A Protein A 7 FT #SUB 14 13 NH2 D 70 93 LYS A Protein B 2 FT #SUB 2 1 THR D 48 71 GLN C Protein B 2 FT #SUB 3 2 SER D 48 71 GLN C Protein A 2 FT #SUB 4 3 PHE D 34 57 GLY C Protein S 1 FT #SUB 4 3 PHE D 37 60 ILE C Protein S 6 FT #SUB 4 3 PHE D 38 61 MET C Protein S 1 FT #SUB 4 3 PHE D 43 66 TYR C Protein S 2 FT #SUB 4 3 PHE D 48 71 GLN C Protein A 5 FT #SUB 4 3 PHE D 69 92 VAL C Protein S 1 FT #SUB 5 4 9E7 D 38 61 MET C Protein S 2 FT #SUB 7 6 TYR D 49 72 HIS C Protein S 11 FT #SUB 7 6 TYR D 69 92 VAL C Protein A 3 FT #SUB 8 7 TRP D 30 53 MET C Protein S 4 FT #SUB 8 7 TRP D 33 56 LEU C Protein S 1 FT #SUB 8 7 TRP D 34 57 GLY C Protein S 7 FT #SUB 8 7 TRP D 69 92 VAL C Protein S 1 FT #SUB 11 10 LEU D 30 53 MET C Protein S 1 FT #SUB 11 10 LEU D 69 92 VAL C Protein S 2 FT #SUB 11 10 LEU D 72 95 PRO C Protein S 1 FT #SUB 11 10 LEU D 76 99 TYR C Protein B 1 FT #SUB 12 11 SER D 30 53 MET C Protein S 3 FT #SUB 13 12 PRO D 27 50 LYS C Protein A 3 FT #SUB 7 6 TYR D 28 51 GLU E Protein S 1 FT #SUB 10 9 LEU D 2 25 ASN E Protein S 1 FT #SUB 10 9 LEU D 3 26 GLN E Protein A 9 CC SEQUENCE 14 AA (ATOM); CC XTSFXEYWCL LSPX CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLLSPX CC ************** SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX // ID 5VK1E STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 20 43 GLN E 70 93 LYS C Protein B 4 FT #SUB 21 44 GLY E 70 93 LYS C Protein B 2 FT #SUB 23 46 MET E 70 93 LYS C Protein B 3 FT #SUB 24 47 PHE E 70 93 LYS C Protein A 7 FT #SUB 28 51 GLU E 70 93 LYS C Protein S 5 FT #SUB 2 25 ASN E 10 9 LEU D Protein S 1 FT #SUB 3 26 GLN E 10 9 LEU D Protein S 9 FT #SUB 28 51 GLU E 7 6 TYR D Protein S 1 FT #SUB 30 53 MET E 8 7 TRP F Protein A 6 FT #SUB 30 53 MET E 11 10 LEU F Protein S 1 FT #SUB 33 56 LEU E 8 7 TRP F Protein A 2 FT #SUB 34 57 GLY E 4 3 PHE F Protein B 1 FT #SUB 34 57 GLY E 8 7 TRP F Protein B 9 FT #SUB 37 60 ILE E 4 3 PHE F Protein S 5 FT #SUB 38 61 MET E 4 3 PHE F Protein S 2 FT #SUB 38 61 MET E 5 4 9E7 F Protein S 1 FT #SUB 43 66 TYR E 4 3 PHE F Protein S 2 FT #SUB 48 71 GLN E 3 2 SER F Protein S 2 FT #SUB 48 71 GLN E 4 3 PHE F Protein A 8 FT #SUB 49 72 HIS E 7 6 TYR F Protein S 2 FT #SUB 51 74 VAL E 4 3 PHE F Protein S 1 FT #SUB 69 92 VAL E 4 3 PHE F Protein S 1 FT #SUB 69 92 VAL E 7 6 TYR F Protein S 2 FT #SUB 69 92 VAL E 8 7 TRP F Protein S 1 FT #SUB 75 98 LEU E 8 7 TRP F Protein S 2 FT #SUB 76 99 TYR E 11 10 LEU F Protein S 1 FT #SUB 20 43 GLN E 20 43 GLN K Protein S 5 FT #SUB 6 29 PRO E 65 88 GLN M Protein B 2 FT #SUB 8 31 LEU E 65 88 GLN M Protein A 7 FT #SUB 11 34 LEU E 52 75 TYR M Protein S 1 FT #SUB 11 34 LEU E 65 88 GLN M Protein S 1 FT #SUB 11 34 LEU E 66 89 SER M Protein S 1 FT #SUB 12 35 LYS E 52 75 TYR M Protein A 4 FT #SUB 15 38 HIS E 50 73 MET M Protein S 2 FT #SUB 15 38 HIS E 52 75 TYR M Protein S 5 FT #SUB 15 38 HIS E 66 89 SER M Protein S 2 FT #SUB 22 45 GLU E 64 87 ARG M Protein S 10 FT #SUB 22 45 GLU E 65 88 GLN M Protein S 6 FT #SUB 22 45 GLU E 66 89 SER M Protein S 2 FT DISORDER 1 1 FT DISORDER 85 85 CC SEQUENCE 83 AA (ATOM); CC NQVRPKLPLL KILHAAGAQG EMFTVKEVMH YLGQYIMVKQ LYDAAAQHMV YCGGDLLGEL CC LGRQSFSVKD PSPLYDMLRK NLV CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM -NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************* CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV- CC ********************************** SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1F STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 3 2 SER F 48 71 GLN E Protein B 2 FT #SUB 4 3 PHE F 34 57 GLY E Protein S 1 FT #SUB 4 3 PHE F 37 60 ILE E Protein S 5 FT #SUB 4 3 PHE F 38 61 MET E Protein S 2 FT #SUB 4 3 PHE F 43 66 TYR E Protein S 2 FT #SUB 4 3 PHE F 48 71 GLN E Protein A 8 FT #SUB 4 3 PHE F 51 74 VAL E Protein S 1 FT #SUB 4 3 PHE F 69 92 VAL E Protein S 1 FT #SUB 5 4 9E7 F 38 61 MET E Protein S 1 FT #SUB 7 6 TYR F 49 72 HIS E Protein S 2 FT #SUB 7 6 TYR F 69 92 VAL E Protein S 2 FT #SUB 8 7 TRP F 30 53 MET E Protein S 6 FT #SUB 8 7 TRP F 33 56 LEU E Protein S 2 FT #SUB 8 7 TRP F 34 57 GLY E Protein S 9 FT #SUB 8 7 TRP F 69 92 VAL E Protein S 1 FT #SUB 8 7 TRP F 75 98 LEU E Protein S 2 FT #SUB 11 10 LEU F 30 53 MET E Protein S 1 FT #SUB 11 10 LEU F 76 99 TYR E Protein S 1 FT DISORDER 12 14 CC SEQUENCE 11 AA (ATOM); CC XTSFXEYWCL L CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLL--- CC *********** SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX // ID 5VK1G STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 39 62 VAL G 7 30 LYS A Protein B 5 FT #SUB 41 64 GLN G 81 104 LYS A Protein S 1 FT #SUB 41 64 GLN G 82 105 ASN A Protein S 3 FT #SUB 45 68 ALA G 60 83 GLU A Protein S 1 FT #SUB 30 53 MET G 8 7 TRP H Protein A 5 FT #SUB 30 53 MET G 11 10 LEU H Protein S 2 FT #SUB 33 56 LEU G 8 7 TRP H Protein S 1 FT #SUB 34 57 GLY G 4 3 PHE H Protein B 2 FT #SUB 34 57 GLY G 8 7 TRP H Protein B 8 FT #SUB 37 60 ILE G 4 3 PHE H Protein S 5 FT #SUB 38 61 MET G 4 3 PHE H Protein S 2 FT #SUB 38 61 MET G 5 4 9E7 H Protein S 1 FT #SUB 43 66 TYR G 4 3 PHE H Protein S 1 FT #SUB 48 71 GLN G 3 2 SER H Protein S 3 FT #SUB 48 71 GLN G 4 3 PHE H Protein A 9 FT #SUB 49 72 HIS G 7 6 TYR H Protein A 9 FT #SUB 69 92 VAL G 4 3 PHE H Protein S 1 FT #SUB 69 92 VAL G 7 6 TYR H Protein S 3 FT #SUB 69 92 VAL G 11 10 LEU H Protein A 2 FT #SUB 72 95 PRO G 11 10 LEU H Protein S 1 FT #SUB 75 98 LEU G 8 7 TRP H Protein S 1 FT #SUB 76 99 TYR G 11 10 LEU H Protein S 2 FT #SUB 20 43 GLN G 5 4 9E7 P Protein S 3 FT #SUB 20 43 GLN G 9 8 CYS P Protein S 3 FT DISORDER 1 1 FT DISORDER 84 85 CC SEQUENCE 82 AA (ATOM); CC NQVRPKLPLL KILHAAGAQG EMFTVKEVMH YLGQYIMVKQ LYDAAAQHMV YCGGDLLGEL CC LGRQSFSVKD PSPLYDMLRK NL CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM -NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************* CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNL-- CC ********************************* SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1H STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 3 2 SER H 48 71 GLN G Protein A 3 FT #SUB 4 3 PHE H 34 57 GLY G Protein S 2 FT #SUB 4 3 PHE H 37 60 ILE G Protein S 5 FT #SUB 4 3 PHE H 38 61 MET G Protein S 2 FT #SUB 4 3 PHE H 43 66 TYR G Protein S 1 FT #SUB 4 3 PHE H 48 71 GLN G Protein A 9 FT #SUB 4 3 PHE H 69 92 VAL G Protein S 1 FT #SUB 5 4 9E7 H 38 61 MET G Protein S 1 FT #SUB 7 6 TYR H 49 72 HIS G Protein S 9 FT #SUB 7 6 TYR H 69 92 VAL G Protein A 3 FT #SUB 8 7 TRP H 30 53 MET G Protein S 5 FT #SUB 8 7 TRP H 33 56 LEU G Protein S 1 FT #SUB 8 7 TRP H 34 57 GLY G Protein S 8 FT #SUB 8 7 TRP H 75 98 LEU G Protein S 1 FT #SUB 11 10 LEU H 30 53 MET G Protein S 2 FT #SUB 11 10 LEU H 69 92 VAL G Protein S 2 FT #SUB 11 10 LEU H 72 95 PRO G Protein S 1 FT #SUB 11 10 LEU H 76 99 TYR G Protein S 2 FT DISORDER 13 14 CC SEQUENCE 12 AA (ATOM); CC XTSFXEYWCL LS CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLLS-- CC ************ SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX // ID 5VK1I STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 26 49 VAL I 2 25 ASN A Protein S 2 FT #SUB 80 103 ARG I 2 25 ASN A Protein S 2 FT #SUB 69 92 VAL I 12 11 SER B Protein B 1 FT #SUB 69 92 VAL I 13 12 PRO B Protein B 1 FT #SUB 70 93 LYS I 9 8 CYS B Protein S 2 FT #SUB 70 93 LYS I 10 9 LEU B Protein S 2 FT #SUB 70 93 LYS I 13 12 PRO B Protein B 5 FT #SUB 72 95 PRO I 13 12 PRO B Protein S 1 FT #SUB 30 53 MET I 8 7 TRP J Protein A 5 FT #SUB 30 53 MET I 12 11 SER J Protein S 4 FT #SUB 33 56 LEU I 8 7 TRP J Protein S 3 FT #SUB 34 57 GLY I 4 3 PHE J Protein B 1 FT #SUB 34 57 GLY I 8 7 TRP J Protein B 6 FT #SUB 37 60 ILE I 4 3 PHE J Protein S 6 FT #SUB 38 61 MET I 4 3 PHE J Protein S 2 FT #SUB 38 61 MET I 5 4 9E7 J Protein S 2 FT #SUB 43 66 TYR I 4 3 PHE J Protein S 3 FT #SUB 48 71 GLN I 2 1 THR J Protein S 2 FT #SUB 48 71 GLN I 3 2 SER J Protein S 4 FT #SUB 48 71 GLN I 4 3 PHE J Protein A 7 FT #SUB 49 72 HIS I 7 6 TYR J Protein A 8 FT #SUB 51 74 VAL I 4 3 PHE J Protein S 1 FT #SUB 69 92 VAL I 4 3 PHE J Protein S 2 FT #SUB 69 92 VAL I 7 6 TYR J Protein S 3 FT #SUB 69 92 VAL I 8 7 TRP J Protein S 3 FT #SUB 69 92 VAL I 11 10 LEU J Protein A 4 FT #SUB 70 93 LYS I 7 6 TYR J Protein S 2 FT #SUB 72 95 PRO I 11 10 LEU J Protein S 2 FT #SUB 75 98 LEU I 8 7 TRP J Protein S 1 FT #SUB 76 99 TYR I 11 10 LEU J Protein S 3 FT #SUB 40 63 LYS I 7 30 LYS M Protein B 2 FT #SUB 41 64 GLN I 7 30 LYS M Protein B 1 FT #SUB 41 64 GLN I 81 104 LYS M Protein S 9 FT #SUB 43 66 TYR I 81 104 LYS M Protein S 3 FT #SUB 44 67 ASP I 60 83 GLU M Protein S 1 FT #SUB 45 68 ALA I 60 83 GLU M Protein S 1 FT #SUB 45 68 ALA I 61 84 LEU M Protein S 1 FT #SUB 45 68 ALA I 62 85 LEU M Protein S 2 FT #SUB 45 68 ALA I 63 86 GLY M Protein A 3 FT #SUB 46 69 ALA I 63 86 GLY M Protein B 1 FT #SUB 20 43 GLN I 70 93 LYS O Protein B 3 FT #SUB 21 44 GLY I 70 93 LYS O Protein B 2 FT #SUB 23 46 MET I 70 93 LYS O Protein B 3 FT #SUB 28 51 GLU I 70 93 LYS O Protein S 2 FT #SUB 28 51 GLU I 7 6 TYR P Protein S 2 FT #SUB 28 51 GLU I 10 9 LEU P Protein S 1 FT DISORDER 1 2 FT DISORDER 85 85 CC SEQUENCE 82 AA (ATOM); CC QVRPKLPLLK ILHAAGAQGE MFTVKEVMHY LGQYIMVKQL YDAAAQHMVY CGGDLLGELL CC GRQSFSVKDP SPLYDMLRKN LV CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM --QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************ CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV- CC ********************************** SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1J STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 9 8 CYS J 76 99 TYR A Protein B 2 FT #SUB 10 9 LEU J 26 49 VAL A Protein B 1 FT #SUB 10 9 LEU J 30 53 MET A Protein S 2 FT #SUB 11 10 LEU J 26 49 VAL A Protein B 4 FT #SUB 13 12 PRO J 26 49 VAL A Protein S 1 FT #SUB 13 12 PRO J 76 99 TYR A Protein A 3 FT #SUB 13 12 PRO J 79 102 LEU A Protein S 1 FT #SUB 14 13 NH2 J 76 99 TYR A Protein B 3 FT #SUB 14 13 NH2 J 80 103 ARG A Protein B 3 FT #SUB 7 6 TYR J 10 9 LEU B Protein S 2 FT #SUB 7 6 TYR J 12 11 SER B Protein A 6 FT #SUB 10 9 LEU J 12 11 SER B Protein S 3 FT #SUB 10 9 LEU J 13 12 PRO B Protein A 3 FT #SUB 11 10 LEU J 12 11 SER B Protein S 2 FT #SUB 11 10 LEU J 13 12 PRO B Protein B 2 FT #SUB 11 10 LEU J 14 13 NH2 B Protein A 2 FT #SUB 5 4 9E7 J 2 25 ASN C Protein S 2 FT #SUB 2 1 THR J 48 71 GLN I Protein B 2 FT #SUB 3 2 SER J 48 71 GLN I Protein A 4 FT #SUB 4 3 PHE J 34 57 GLY I Protein S 1 FT #SUB 4 3 PHE J 37 60 ILE I Protein S 6 FT #SUB 4 3 PHE J 38 61 MET I Protein S 2 FT #SUB 4 3 PHE J 43 66 TYR I Protein S 3 FT #SUB 4 3 PHE J 48 71 GLN I Protein A 7 FT #SUB 4 3 PHE J 51 74 VAL I Protein S 1 FT #SUB 4 3 PHE J 69 92 VAL I Protein S 2 FT #SUB 5 4 9E7 J 38 61 MET I Protein S 2 FT #SUB 7 6 TYR J 49 72 HIS I Protein S 8 FT #SUB 7 6 TYR J 69 92 VAL I Protein A 3 FT #SUB 7 6 TYR J 70 93 LYS I Protein S 2 FT #SUB 8 7 TRP J 30 53 MET I Protein S 5 FT #SUB 8 7 TRP J 33 56 LEU I Protein S 3 FT #SUB 8 7 TRP J 34 57 GLY I Protein S 6 FT #SUB 8 7 TRP J 69 92 VAL I Protein A 3 FT #SUB 8 7 TRP J 75 98 LEU I Protein S 1 FT #SUB 11 10 LEU J 69 92 VAL I Protein S 4 FT #SUB 11 10 LEU J 72 95 PRO I Protein S 2 FT #SUB 11 10 LEU J 76 99 TYR I Protein A 3 FT #SUB 12 11 SER J 30 53 MET I Protein S 4 CC SEQUENCE 14 AA (ATOM); CC XTSFXEYWCL LSPX CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLLSPX CC ************** SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX // ID 5VK1K STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 6 29 PRO K 65 88 GLN C Protein B 3 FT #SUB 7 30 LYS K 65 88 GLN C Protein B 2 FT #SUB 8 31 LEU K 52 75 TYR C Protein S 2 FT #SUB 8 31 LEU K 54 77 GLY C Protein S 2 FT #SUB 8 31 LEU K 55 78 GLY C Protein S 1 FT #SUB 8 31 LEU K 65 88 GLN C Protein A 4 FT #SUB 11 34 LEU K 66 89 SER C Protein S 2 FT #SUB 12 35 LYS K 52 75 TYR C Protein B 1 FT #SUB 15 38 HIS K 50 73 MET C Protein S 2 FT #SUB 15 38 HIS K 52 75 TYR C Protein S 4 FT #SUB 15 38 HIS K 66 89 SER C Protein S 1 FT #SUB 22 45 GLU K 64 87 ARG C Protein S 16 FT #SUB 22 45 GLU K 65 88 GLN C Protein S 1 FT #SUB 22 45 GLU K 66 89 SER C Protein S 3 FT #SUB 20 43 GLN K 20 43 GLN E Protein S 5 FT #SUB 30 53 MET K 8 7 TRP L Protein A 6 FT #SUB 33 56 LEU K 8 7 TRP L Protein S 1 FT #SUB 34 57 GLY K 4 3 PHE L Protein B 1 FT #SUB 34 57 GLY K 8 7 TRP L Protein B 8 FT #SUB 37 60 ILE K 4 3 PHE L Protein S 5 FT #SUB 37 60 ILE K 8 7 TRP L Protein S 1 FT #SUB 38 61 MET K 4 3 PHE L Protein S 2 FT #SUB 38 61 MET K 5 4 9E7 L Protein S 1 FT #SUB 43 66 TYR K 4 3 PHE L Protein S 4 FT #SUB 48 71 GLN K 2 1 THR L Protein S 2 FT #SUB 48 71 GLN K 3 2 SER L Protein S 7 FT #SUB 48 71 GLN K 4 3 PHE L Protein A 8 FT #SUB 49 72 HIS K 7 6 TYR L Protein A 5 FT #SUB 69 92 VAL K 4 3 PHE L Protein S 2 FT #SUB 69 92 VAL K 7 6 TYR L Protein S 3 FT #SUB 69 92 VAL K 8 7 TRP L Protein S 2 FT #SUB 69 92 VAL K 11 10 LEU L Protein A 2 FT #SUB 72 95 PRO K 11 10 LEU L Protein S 1 FT #SUB 75 98 LEU K 8 7 TRP L Protein S 1 FT #SUB 20 43 GLN K 70 93 LYS M Protein B 3 FT #SUB 21 44 GLY K 70 93 LYS M Protein B 1 FT #SUB 23 46 MET K 70 93 LYS M Protein B 2 FT #SUB 24 47 PHE K 70 93 LYS M Protein S 2 FT #SUB 28 51 GLU K 70 93 LYS M Protein S 4 FT #SUB 3 26 GLN K 10 9 LEU N Protein B 1 FT #SUB 27 50 LYS K 1 0 ACE N Protein S 1 FT #SUB 27 50 LYS K 2 1 THR N Protein S 2 FT #SUB 28 51 GLU K 7 6 TYR N Protein S 2 FT DISORDER 1 2 FT DISORDER 85 85 CC SEQUENCE 82 AA (ATOM); CC QVRPKLPLLK ILHAAGAQGE MFTVKEVMHY LGQYIMVKQL YDAAAQHMVY CGGDLLGELL CC GRQSFSVKDP SPLYDMLRKN LV CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM --QVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************ CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLV- CC ********************************** SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1L STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 2 1 THR L 48 71 GLN K Protein B 2 FT #SUB 3 2 SER L 48 71 GLN K Protein A 7 FT #SUB 4 3 PHE L 34 57 GLY K Protein S 1 FT #SUB 4 3 PHE L 37 60 ILE K Protein S 5 FT #SUB 4 3 PHE L 38 61 MET K Protein S 2 FT #SUB 4 3 PHE L 43 66 TYR K Protein S 4 FT #SUB 4 3 PHE L 48 71 GLN K Protein A 8 FT #SUB 4 3 PHE L 69 92 VAL K Protein S 2 FT #SUB 5 4 9E7 L 38 61 MET K Protein S 1 FT #SUB 7 6 TYR L 49 72 HIS K Protein S 5 FT #SUB 7 6 TYR L 69 92 VAL K Protein A 3 FT #SUB 8 7 TRP L 30 53 MET K Protein S 6 FT #SUB 8 7 TRP L 33 56 LEU K Protein S 1 FT #SUB 8 7 TRP L 34 57 GLY K Protein S 8 FT #SUB 8 7 TRP L 37 60 ILE K Protein S 1 FT #SUB 8 7 TRP L 69 92 VAL K Protein B 2 FT #SUB 8 7 TRP L 75 98 LEU K Protein S 1 FT #SUB 11 10 LEU L 69 92 VAL K Protein S 2 FT #SUB 11 10 LEU L 72 95 PRO K Protein S 1 FT DISORDER 13 14 CC SEQUENCE 12 AA (ATOM); CC XTSFXEYWCL LS CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLLS-- CC ************ SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX // ID 5VK1M STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 64 87 ARG M 71 94 ASP C Protein S 2 FT #SUB 71 94 ASP M 64 87 ARG C Protein S 1 FT #SUB 71 94 ASP M 71 94 ASP C Protein S 3 FT #SUB 73 96 SER M 64 87 ARG C Protein S 1 FT #SUB 73 96 SER M 73 96 SER C Protein A 3 FT #SUB 73 96 SER M 74 97 PRO C Protein S 1 FT #SUB 74 97 PRO M 71 94 ASP C Protein S 1 FT #SUB 74 97 PRO M 73 96 SER C Protein B 2 FT #SUB 80 103 ARG M 80 103 ARG C Protein S 11 FT #SUB 50 73 MET M 15 38 HIS E Protein S 2 FT #SUB 52 75 TYR M 11 34 LEU E Protein S 1 FT #SUB 52 75 TYR M 12 35 LYS E Protein S 4 FT #SUB 52 75 TYR M 15 38 HIS E Protein S 5 FT #SUB 64 87 ARG M 22 45 GLU E Protein A 10 FT #SUB 65 88 GLN M 6 29 PRO E Protein S 2 FT #SUB 65 88 GLN M 8 31 LEU E Protein A 7 FT #SUB 65 88 GLN M 11 34 LEU E Protein S 1 FT #SUB 65 88 GLN M 22 45 GLU E Protein A 6 FT #SUB 66 89 SER M 11 34 LEU E Protein S 1 FT #SUB 66 89 SER M 15 38 HIS E Protein S 2 FT #SUB 66 89 SER M 22 45 GLU E Protein B 2 FT #SUB 7 30 LYS M 40 63 LYS I Protein S 2 FT #SUB 7 30 LYS M 41 64 GLN I Protein S 1 FT #SUB 60 83 GLU M 44 67 ASP I Protein B 1 FT #SUB 60 83 GLU M 45 68 ALA I Protein B 1 FT #SUB 61 84 LEU M 45 68 ALA I Protein B 1 FT #SUB 62 85 LEU M 45 68 ALA I Protein B 2 FT #SUB 63 86 GLY M 45 68 ALA I Protein B 3 FT #SUB 63 86 GLY M 46 69 ALA I Protein B 1 FT #SUB 81 104 LYS M 41 64 GLN I Protein A 9 FT #SUB 81 104 LYS M 43 66 TYR I Protein S 3 FT #SUB 70 93 LYS M 20 43 GLN K Protein S 3 FT #SUB 70 93 LYS M 21 44 GLY K Protein S 1 FT #SUB 70 93 LYS M 23 46 MET K Protein S 2 FT #SUB 70 93 LYS M 24 47 PHE K Protein S 2 FT #SUB 70 93 LYS M 28 51 GLU K Protein S 4 FT #SUB 30 53 MET M 8 7 TRP N Protein A 5 FT #SUB 30 53 MET M 11 10 LEU N Protein S 1 FT #SUB 33 56 LEU M 8 7 TRP N Protein S 2 FT #SUB 34 57 GLY M 4 3 PHE N Protein B 1 FT #SUB 34 57 GLY M 8 7 TRP N Protein B 8 FT #SUB 37 60 ILE M 4 3 PHE N Protein S 4 FT #SUB 38 61 MET M 4 3 PHE N Protein S 2 FT #SUB 38 61 MET M 5 4 9E7 N Protein S 1 FT #SUB 43 66 TYR M 4 3 PHE N Protein S 7 FT #SUB 48 71 GLN M 2 1 THR N Protein S 2 FT #SUB 48 71 GLN M 3 2 SER N Protein S 4 FT #SUB 48 71 GLN M 4 3 PHE N Protein A 6 FT #SUB 48 71 GLN M 7 6 TYR N Protein B 1 FT #SUB 49 72 HIS M 7 6 TYR N Protein A 9 FT #SUB 69 92 VAL M 4 3 PHE N Protein S 1 FT #SUB 69 92 VAL M 7 6 TYR N Protein S 2 FT #SUB 69 92 VAL M 8 7 TRP N Protein S 1 FT #SUB 69 92 VAL M 11 10 LEU N Protein A 2 FT #SUB 72 95 PRO M 11 10 LEU N Protein S 1 FT #SUB 75 98 LEU M 8 7 TRP N Protein S 1 FT #SUB 76 99 TYR M 11 10 LEU N Protein S 1 FT DISORDER 1 1 FT DISORDER 84 85 CC SEQUENCE 82 AA (ATOM); CC NQVRPKLPLL KILHAAGAQG EMFTVKEVMH YLGQYIMVKQ LYDAAAQHMV YCGGDLLGEL CC LGRQSFSVKD PSPLYDMLRK NL CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM -NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************* CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNL-- CC ********************************* SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1N STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 1 0 ACE N 27 50 LYS K Protein S 1 FT #SUB 2 1 THR N 27 50 LYS K Protein A 2 FT #SUB 7 6 TYR N 28 51 GLU K Protein S 2 FT #SUB 10 9 LEU N 3 26 GLN K Protein B 1 FT #SUB 2 1 THR N 48 71 GLN M Protein B 2 FT #SUB 3 2 SER N 48 71 GLN M Protein A 4 FT #SUB 4 3 PHE N 34 57 GLY M Protein S 1 FT #SUB 4 3 PHE N 37 60 ILE M Protein S 4 FT #SUB 4 3 PHE N 38 61 MET M Protein S 2 FT #SUB 4 3 PHE N 43 66 TYR M Protein S 7 FT #SUB 4 3 PHE N 48 71 GLN M Protein A 6 FT #SUB 4 3 PHE N 69 92 VAL M Protein S 1 FT #SUB 5 4 9E7 N 38 61 MET M Protein S 1 FT #SUB 7 6 TYR N 48 71 GLN M Protein S 1 FT #SUB 7 6 TYR N 49 72 HIS M Protein S 9 FT #SUB 7 6 TYR N 69 92 VAL M Protein B 2 FT #SUB 8 7 TRP N 30 53 MET M Protein S 5 FT #SUB 8 7 TRP N 33 56 LEU M Protein S 2 FT #SUB 8 7 TRP N 34 57 GLY M Protein S 8 FT #SUB 8 7 TRP N 69 92 VAL M Protein S 1 FT #SUB 8 7 TRP N 75 98 LEU M Protein S 1 FT #SUB 11 10 LEU N 30 53 MET M Protein S 1 FT #SUB 11 10 LEU N 69 92 VAL M Protein S 2 FT #SUB 11 10 LEU N 72 95 PRO M Protein S 1 FT #SUB 11 10 LEU N 76 99 TYR M Protein S 1 FT DISORDER 13 14 CC SEQUENCE 12 AA (ATOM); CC XTSFXEYWCL LS CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLLS-- CC ************ SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX // ID 5VK1O STANDARD; PRT; 85 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Protein Mdm4 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 70 93 LYS O 20 43 GLN I Protein S 3 FT #SUB 70 93 LYS O 21 44 GLY I Protein A 2 FT #SUB 70 93 LYS O 23 46 MET I Protein S 3 FT #SUB 70 93 LYS O 28 51 GLU I Protein S 2 FT #SUB 30 53 MET O 8 7 TRP P Protein A 5 FT #SUB 30 53 MET O 11 10 LEU P Protein S 1 FT #SUB 34 57 GLY O 4 3 PHE P Protein B 1 FT #SUB 34 57 GLY O 8 7 TRP P Protein B 7 FT #SUB 37 60 ILE O 4 3 PHE P Protein S 4 FT #SUB 37 60 ILE O 8 7 TRP P Protein S 2 FT #SUB 38 61 MET O 5 4 9E7 P Protein S 2 FT #SUB 43 66 TYR O 4 3 PHE P Protein S 1 FT #SUB 48 71 GLN O 2 1 THR P Protein S 1 FT #SUB 48 71 GLN O 3 2 SER P Protein S 3 FT #SUB 48 71 GLN O 4 3 PHE P Protein A 7 FT #SUB 49 72 HIS O 7 6 TYR P Protein A 4 FT #SUB 51 74 VAL O 4 3 PHE P Protein S 1 FT #SUB 69 92 VAL O 4 3 PHE P Protein S 1 FT #SUB 69 92 VAL O 8 7 TRP P Protein S 1 FT #SUB 69 92 VAL O 11 10 LEU P Protein S 1 FT #SUB 72 95 PRO O 11 10 LEU P Protein S 2 FT #SUB 76 99 TYR O 11 10 LEU P Protein S 2 FT DISORDER 1 1 FT DISORDER 84 85 CC SEQUENCE 82 AA (ATOM); CC NQVRPKLPLL KILHAAGAQG EMFTVKEVMH YLGQYIMVKQ LYDAAAQHMV YCGGDLLGEL CC LGRQSFSVKD PSPLYDMLRK NL CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES INQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ATOM -NQVRPKLPLLKILHAAGAQGEMFTVKEVMHYLGQYIMVKQLYDAAAQHM CC ************************************************* CC SEQRES VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNLVT CC ATOM VYCGGDLLGELLGRQSFSVKDPSPLYDMLRKNL-- CC ********************************* SQ SEQUENCE 85 AA; MW; CN; INQVRPKLPL LKILHAAGAQ GEMFTVKEVM HYLGQYIMVK QLYDAAAQHM VYCGGDLLGE LLGRQSFSVK DPSPLYDMLR KNLVT // ID 5VK1P STANDARD; PRT; 14 AA. DT CONVERTED FROM PDB (SEQRES) 5VK1 DE Lysine-cysteine side chain dithiocarbamate stapled peptide inhibitor PMI OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.690 CC R-Factor 0.281 FT #SUB 5 4 9E7 P 20 43 GLN G Protein S 3 FT #SUB 9 8 CYS P 20 43 GLN G Protein S 3 FT #SUB 7 6 TYR P 28 51 GLU I Protein S 2 FT #SUB 10 9 LEU P 28 51 GLU I Protein S 1 FT #SUB 2 1 THR P 48 71 GLN O Protein B 1 FT #SUB 3 2 SER P 48 71 GLN O Protein A 3 FT #SUB 4 3 PHE P 34 57 GLY O Protein S 1 FT #SUB 4 3 PHE P 37 60 ILE O Protein S 4 FT #SUB 4 3 PHE P 43 66 TYR O Protein S 1 FT #SUB 4 3 PHE P 48 71 GLN O Protein A 7 FT #SUB 4 3 PHE P 51 74 VAL O Protein S 1 FT #SUB 4 3 PHE P 69 92 VAL O Protein S 1 FT #SUB 5 4 9E7 P 38 61 MET O Protein S 2 FT #SUB 7 6 TYR P 49 72 HIS O Protein S 4 FT #SUB 8 7 TRP P 30 53 MET O Protein S 5 FT #SUB 8 7 TRP P 34 57 GLY O Protein S 7 FT #SUB 8 7 TRP P 37 60 ILE O Protein S 2 FT #SUB 8 7 TRP P 69 92 VAL O Protein S 1 FT #SUB 11 10 LEU P 30 53 MET O Protein S 1 FT #SUB 11 10 LEU P 69 92 VAL O Protein S 1 FT #SUB 11 10 LEU P 72 95 PRO O Protein S 2 FT #SUB 11 10 LEU P 76 99 TYR O Protein S 2 FT DISORDER 12 14 CC SEQUENCE 11 AA (ATOM); CC XTSFXEYWCL L CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XTSFXEYWCLLSPX CC ATOM XTSFXEYWCLL--- CC *********** SQ SEQUENCE 14 AA; MW; CN; XTSFXEYWCL LSPX //