1 DJZ 3,5-dimethyl-4-{[2-({1-[4-(methylsulfonyl)benzyl]piperidin-4-yl}amino)pyrimidin-4-yl]oxy}benzonitrile 1.000 2 K5A 4-[(4-{[4-(4-cyano-2,6-dimethylphenoxy)thieno[3,2-D]pyrimidin-2-yl]amino}piperidin-1-yl)methyl]benzene-1-sulfonamide 0.872 3 WB3 (2e)-3-[4-({2-[(1-{[4-(methanesulfonyl)phenyl]methyl}piperidin-4-yl)amino]pyrido[2,3-D]pyrimidin-4-yl}oxy)-3,5-dimethylphenyl]prop-2-enenitrile 0.810 4 K5C 4-({4-[(4-{4-[(E)-2-cyanoethenyl]-2,6-dimethylphenoxy}thieno[3,2-D]pyrimidin-2-yl)amino]piperidin-1-yl}methyl)benzene-1-sulfonamide 0.786 5 K7F 4-[(4-{[4-(4-cyano-2,6-dimethylphenoxy)-5-(pyridin-4-yl)pyrimidin-2-yl]amino}piperidin-1-yl)methyl]benzamide 0.705