1 BHV Tert-butyl 4-(2-{3-[3-{[(3-methylbut-2-enoyl)amino]methyl}-4-(trifluoromethyl)phenyl]-1-[3-(morpholin-4-yl)propyl]-1,4,6,7-tetrahydro-5h-pyrazolo[4,3-C]pyridin-5-yl}-2-oxoethyl)piperidine-1-carboxylate 1.000 2 BGY Tert-butyl 4-(2-{3-(4-chloro-3-iodophenyl)-1-[3-(morpholin-4-yl)propyl]-1,4,6,7-tetrahydro-5h-pyrazolo[4,3-C]pyridin-5-yl}-2-oxoethyl)piperidine-1-carboxylate 0.741 3 BG7 N-{[5-{1-[3-(dimethylamino)propyl]-5-[(piperidin-4-yl)acetyl]-4,5,6,7-tetrahydro-1h-pyrazolo[4,3-C]pyridin-3-yl}-2-(trifluoromethyl)phenyl]methyl}-3-methylbut-2-enamide 0.709