1 B4Y (2r)-N-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide 1.000 2 B5G (2r)-N-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-C]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide 0.846