1 8DV (R)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholine 1.000 2 VCD 4-{4-[(3r)-3-methylmorpholin-4-yl]-6-[1-(methylsulfonyl)cyclopropyl]pyrimidin-2-yl}-1h-indole 0.875 3 XXV 1-{6-[(3r)-3-methylmorpholin-4-yl]-2-(1h-pyrrolo[2,3-B]pyridin-4-yl)pyrimidin-4-yl}cyclopropane-1-sulfonamide 0.818 4 VJM 4-(4-{1-[(R)-amino(hydroxy)methyl-lambda~4~-sulfanyl]cyclopropyl}-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-2-yl)-1h-pyrrolo[2,3-B]pyridine 0.765 5 XXS 4-{4-[(3r)-3-methylmorpholin-4-yl]-6-[1-(S-methylsulfonimidoyl)cyclopropyl]pyrimidin-2-yl}-1h-indazole 0.765 6 XWV 5-{4-[(3r)-3-methylmorpholin-4-yl]-6-[1-(S-methylsulfonimidoyl)cyclopropyl]pyrimidin-2-yl}isoquinoline 0.743 7 XWY (3r)-3-methyl-4-{6-[1-(S-methylsulfonimidoyl)cyclopropyl]-2-(naphthalen-1-yl)pyrimidin-4-yl}morpholine 0.743 8 VQS N-(4-{4-[1-(cyclopropylsulfonyl)cyclopropyl]-6-[(3s)-3-methylmorpholin-4-yl]pyrimidin-2-yl}phenyl)-N'-(2-hydroxyethyl)thiourea 0.737