PDB ID: 6K04
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CQF | (6~{R})-~{N}-(4-chlorophenyl)-1-methyl-8-(1-methylpyrazol-4-yl)-5,6-dihydro-4~{H}-[1,2,4]triazolo[4,3-a][1]benzazepin-6-amine | PoSSuM |
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Download interaction data: 6K04
Structure summary
Code : | 6K04 PDBj RCSB PDB PDBe | ||||||||||||
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Header : | ANTITUMOR PROTEIN | ||||||||||||
Title : | Crystal structure of BRD2(BD2)with ligand BY27 bound | ||||||||||||
Release Data : | 2019-09-18 | ||||||||||||
Compound : |
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Authors : | Lu, T., Lu, W., Chen, D., Zhao, Y., Luo, C. | ||||||||||||
Keywords : | Antitumor; BET proteins; Bromodomain inhibitor; Epigenetic readers, ANTITUMOR PROTEIN | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.251 Å ) | ||||||||||||
Citation : |
Discovery, structural insight, and bioactivities of BY27 as a selective inhibitor of the second bromodomains of BET proteins.
Chen, D.,Lu, T.,Yan, Z.
et al.
PubMed: 31461688 |
Reaction
Chain : | A |
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UniProt : | P25440 (BRD2_HUMAN) |
Reaction : | - |