PDB ID: 6GVA
Hetero Atom Contents
The number of atoms exceeds 100,000. So, it can not be displayed here.
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Data format:
Color scheme of protein:
Code | Name | Style | Show | Link | |
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BR | Bromide ion | PoSSuM | |||
CL | Chloride ion | PoSSuM | |||
EDO | 1,2-ethanediol | PoSSuM | |||
FCQ | 5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{N}-[(4-pyridin-2-ylphenyl)methyl]-2~{H}-pyrazolo[4,3-D]pyrimidin-7-amine | PoSSuM | |||
PG4 | Tetraethylene glycol | PoSSuM | |||
PGE | Triethylene glycol | PoSSuM | |||
SGM | Monothioglycerol | PoSSuM |
Code | Name | Show |
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TPO | Phosphothreonine |
Code | Name | Emphasize |
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Code | Name | Show |
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Download interaction data: 6GVA
Structure summary
Code : | 6GVA PDBj RCSB PDB PDBe | ||||||||||||||||||||||||
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Header : | CELL CYCLE | ||||||||||||||||||||||||
Title : | CDK2/cyclin A2 in complex with pyrazolo[4,3-D]pyrimidine inhibitor LGR4455 | ||||||||||||||||||||||||
Release Data : | 2019-05-01 | ||||||||||||||||||||||||
Compound : |
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Source : |
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Authors : | Skerlova, J., Rezacova, P. | ||||||||||||||||||||||||
Keywords : | cyclin-dependent kinase, pyrazolo[4, 3-d]pyrimidine, CELL CYCLE | ||||||||||||||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.1500 Å ) | ||||||||||||||||||||||||
Citation : |
3,5,7-Substituted Pyrazolo[4,3- d]pyrimidine Inhibitors of Cyclin-Dependent Kinases and Their Evaluation in Lymphoma Models.
Jorda, R.,Havlicek, L.,Sturc, A.
et al.
PubMed: 30943029 |
Reaction
Chain : | A | ||||||||||||
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UniProt : | P24941 (CDK2_HUMAN) | ||||||||||||
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Chain : | B |
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UniProt : | P20248 (CCNA2_HUMAN) |
Reaction : | - |