PDB ID: 6Q8K
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Structure summary
Code : | 6Q8K PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE | ||||||||||||
Title : | CLK1 with bound pyridoquinazoline | ||||||||||||
Release Data : | 2019-02-20 | ||||||||||||
Compound : |
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Source : |
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Authors : | Schroeder, M., Tazarki, H., Zeinyeh, W., Esvan, Y.J., Khiari, J., Joesselin, B., Bach, S., Ruchaud, S., Anizon, F., Giraud, F., Moreau, P., Arrowsmith, C.H., Edwards, A.M., Bountra, C., Knapp, S., Structural Genomics Consortium (SGC) | ||||||||||||
Keywords : | CLK1, Dual specifity protein kinase CLK1, Inhibitor, Kinase, Structural Genomics, Structural Genomics Consortium, SGC, TRANSFERASE | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.29 Å ) | ||||||||||||
Citation : |
New pyrido[3,4-g]quinazoline derivatives as CLK1 and DYRK1A inhibitors: synthesis, biological evaluation and binding mode analysis.
Tazarki, H.,Zeinyeh, W.,Esvan, Y.J.
et al.
PubMed: 30731399 |
Reaction
Chain : | A | ||||||||||||||||
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UniProt : | P49759 (CLK1_HUMAN) | ||||||||||||||||
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