PDB ID: 6PS2
Hetero Atom Contents
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Code | Name | Style | Show | Link | |
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CLR | Cholesterol | PoSSuM | |||
JTZ | (2s)-1-[(1-methylethyl)amino]-3-(2-prop-2-en-1-ylphenoxy)propan-2-ol | PoSSuM | |||
OLA | Oleic acid | PoSSuM | |||
OLB | (2s)-2,3-dihydroxypropyl (9z)-octadec-9-enoate | PoSSuM | |||
OLC | (2r)-2,3-dihydroxypropyl (9z)-octadec-9-enoate | PoSSuM | |||
SO4 | Sulfate ion | PoSSuM |
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Download interaction data: 6PS2
Structure summary
Code : | 6PS2 PDBj RCSB PDB PDBe | ||||||||||||
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Header : | MEMBRANE PROTEIN | ||||||||||||
Title : | XFEL beta2 AR structure by ligand exchange from Timolol to Alprenolol. | ||||||||||||
Release Data : | 2019-11-13 | ||||||||||||
Compound : |
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Authors : | Ishchenko, A., Stauch, B., Han, G.W., Batyuk, A., Shiriaeva, A., Li, C., Zatsepin, N.A., Weierstall, U., Liu, W., Nango, E., Nakane, T., Tanaka, R., Tono, K., Joti, Y., Iwata, S., Moraes, I., Gati, C., Cherezov, C. | ||||||||||||
Keywords : | GPCR, COMPLEX-LCP method, SBDD, drug design, XFEL, LCP-SFX, Ligand Exchange, Timolol, Alprenolol, MEMBRANE PROTEIN, b2AR, beta2AR | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.4000 Å ) | ||||||||||||
Citation : |
Toward G protein-coupled receptor structure-based drug design using X-ray lasers.
Ishchenko, A.,Stauch, B.,Han, G.W.
et al.
PubMed: 31709066 |
Reaction
Chain : | A |
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UniProt : | P07550 (ADRB2_HUMAN) |
Reaction : | - |
Chain : | A | ||||||||
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UniProt : | D9IEF7 (D9IEF7_BPT4) | ||||||||
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