PDB ID: 6EGA
Hetero Atom Contents
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Code | Name | Style | Show | Link | |
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J8A | 3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-B]pyridin-5-yl}-N-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | PoSSuM | |||
SO4 | Sulfate ion | PoSSuM | |||
CO | Cobalt (II) ion | PoSSuM |
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Download interaction data: 6EGA
Structure summary
Code : | 6EGA PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | IRAK4 in complex with a type II inhibitor | ||||||||||||
Release Data : | 2019-02-20 | ||||||||||||
Compound : |
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Source : |
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Authors : | Wang, L., Wu, H. | ||||||||||||
Keywords : | Inhibitor, Complex, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.512 Å ) | ||||||||||||
Citation : |
Conformational flexibility and inhibitor binding to unphosphorylated interleukin-1 receptor-associated kinase 4 (IRAK4).
Wang, L.,Ferrao, R.,Li, Q.
et al.
PubMed: 30679311 |
Reaction
Chain : | A, B | ||||||||||||
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UniProt : | Q9NWZ3 (IRAK4_HUMAN) | ||||||||||||
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