PDB ID: 6B3E
Hetero Atom Contents
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Color scheme of protein:
Code | Name | Style | Show | Link | |
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MG | Magnesium ion | PoSSuM | |||
CJM | 2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-ol | PoSSuM | |||
EDO | 1,2-ethanediol | PoSSuM |
Code | Name | Show |
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TPO | Phosphothreonine |
Code | Name | Emphasize |
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Code | Name | Show |
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Download interaction data: 6B3E
Structure summary
Code : | 6B3E PDBj RCSB PDB PDBe | ||||||||||||||||||||||||
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Header : | TRANSFERASE/INHIBITOR | ||||||||||||||||||||||||
Title : | Crystal structure of human CDK12/CyclinK in complex with an inhibitor | ||||||||||||||||||||||||
Release Data : | 2017-12-27 | ||||||||||||||||||||||||
Compound : |
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Source : |
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Authors : | Ferguson, A.D. | ||||||||||||||||||||||||
Keywords : | Inhibitor, complex, kinase, TRANSFERASE, TRANSFERASE-INHIBITOR complex | ||||||||||||||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 3.06 Å ) | ||||||||||||||||||||||||
Citation : |
Structure-Based Design of Selective Noncovalent CDK12 Inhibitors.
Johannes, J.W.,Denz, C.R.,Su, N.
et al.
PubMed: 29266803 |
Reaction
Chain : | A, C | ||||||||||||||||
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UniProt : | Q9NYV4 (CDK12_HUMAN) | ||||||||||||||||
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Chain : | B, D |
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UniProt : | O75909 (CCNK_HUMAN) |
Reaction : | - |