PDB ID: 5W9D
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Structure summary
Code : | 5W9D PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSCRIPTION | ||||||||||||
Title : | Estrogen Receptor Alpha Ligand Binding Domain C381S, C417S, C530S Mutant in Complex with Endoxifen | ||||||||||||
Release Data : | 2017-10-11 | ||||||||||||
Compound : |
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Source : |
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Authors : | Fanning, S.W., Greene, G.L. | ||||||||||||
Keywords : | Breast Cancer, Selective Estrogen Receptor Modulator, TRANSCRIPTION | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.6464 Å ) | ||||||||||||
Citation : |
Endoxifen, 4-Hydroxytamoxifen and an Estrogenic Derivative Modulate Estrogen Receptor Complex Mediated Apoptosis in Breast Cancer.
Maximov, P.Y.,Abderrahman, B.,Fanning, S.W.
et al.
PubMed: 29739819 |
Reaction
Chain : | A, B |
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UniProt : | P03372 (ESR1_HUMAN) |
Reaction : | - |