PDB ID: 5WYX
Hetero Atom Contents
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Data format:
Color scheme of protein:
Code | Name | Style | Show | Link | |
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CU8 | 7-(3-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | PoSSuM |
Code | Name | Show |
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Code | Name | Emphasize |
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BMA | Beta-D-mannopyranose | |
MAN | Alpha-D-mannopyranose | |
NAG | 2-acetamido-2-deoxy-beta-D-glucopyranose |
Code | Name | Show |
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Download interaction data: 5WYX
Structure summary
Code : | 5WYX PDBj RCSB PDB PDBe | ||||||||||||
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Header : | IMMUNE SYSTEM | ||||||||||||
Title : | Crystal structure of human TLR8 in complex with CU-CPT8m | ||||||||||||
Release Data : | 2017-12-13 | ||||||||||||
Compound : |
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Source : |
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Authors : | Tanji, H., Ohto, U., Shimizu, T. | ||||||||||||
Keywords : | IMMUNE SYSTEM | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.40 Å ) | ||||||||||||
Citation : |
Small-molecule inhibition of TLR8 through stabilization of its resting state
Zhang, S.,Hu, Z.,Tanji, H.
et al.
PubMed: 29155428 |
Reaction
Chain : | A, B |
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UniProt : | Q9NR97 (TLR8_HUMAN) |
Reaction : | - |