PDB ID: 5VOM
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Structure summary
Code : | 5VOM PDBj RCSB PDB PDBe | ||||||||||||
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Header : | Transcription/Inhibitor | ||||||||||||
Title : | Benzopiperazine BET bromodomain inhibitor in complex with BD1 of Brd4 | ||||||||||||
Release Data : | 2017-08-02 | ||||||||||||
Compound : |
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Source : |
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Authors : | Toms, A.V., Herbertz, T. | ||||||||||||
Keywords : | bromodomain Brd4 BET Benzopiperazine, Transcription-Inhibitor complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.67 Å ) | ||||||||||||
Citation : |
Design and Optimization of Benzopiperazines as Potent Inhibitors of BET Bromodomains.
Millan, D.S.,Kayser-Bricker, K.J.,Martin, M.W.
et al.
PubMed: 28835800 |
Reaction
Chain : | A, B |
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UniProt : | O60885 (BRD4_HUMAN) |
Reaction : | - |