PDB ID: 5VCW
Hetero Atom Contents
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93J | (2e)-N-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide | PoSSuM | |||
SO4 | Sulfate ion | PoSSuM | |||
EDO | 1,2-ethanediol | PoSSuM |
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Download interaction data: 5VCW
Structure summary
Code : | 5VCW PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | CRYSTAL STRUCTURE OF HUMAN MYT1 KINASE DOMAIN IN COMPLEX WITH Pelitinib | ||||||||||||
Release Data : | 2017-08-23 | ||||||||||||
Compound : |
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Source : |
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Authors : | Zhu, J.-Y., Schonbrunn, E. | ||||||||||||
Keywords : | KINASE DOMAIN, CELL CYCLE, TYROSINE- AND THREONINE-SPECIFIC KINASE, MEMBRANE-ASSOCIATED PROTEIN KINASE, TRANSFERASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.2500 Å ) | ||||||||||||
Citation : |
Structural Basis of Wee Kinases Functionality and Inactivation by Diverse Small Molecule Inhibitors.
Zhu, J.Y.,Cuellar, R.A.,Berndt, N.
et al.
PubMed: 28792760 |
Reaction
Chain : | A, B | ||||||||||||
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UniProt : | Q99640 (PMYT1_HUMAN) | ||||||||||||
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