PDB ID: 5V80
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Structure summary
Code : | 5V80 PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/INHIBITOR | ||||||||||||
Title : | PIM1 kinase in complex with Cpd1 (1-methyl-4-(3-(6-(piperazin-1-yl)pyridin-2-yl)-1H-pyrazolo[3,4-C]pyridin-5-yl)piperazin-2-one) | ||||||||||||
Release Data : | 2018-04-18 | ||||||||||||
Compound : |
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Source : |
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Authors : | Murray, J.M., Wallweber, H. | ||||||||||||
Keywords : | PIM1, SBDD, TRANSFERASE-INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.2520 Å ) | ||||||||||||
Citation : |
Discovery of 5-Azaindazole (GNE-955) as a Potent Pan-Pim Inhibitor with Optimized Bioavailability.
Wang, X.,Kolesnikov, A.,Tay, S.
et al.
PubMed: 28445037 |
Reaction
Chain : | A | ||||||||||||
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UniProt : | P11309 (PIM1_HUMAN) | ||||||||||||
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