PDB ID: 5V61
Hetero Atom Contents
The number of atoms exceeds 100,000. So, it can not be displayed here.
Select unit:
Select hetatm:
Select chain: Sequence
Data format:
Color scheme of protein:
Code | Name | Style | Show | Link | |
---|---|---|---|---|---|
90A | 2-oxo-6,9,12,15-tetraoxa-3-azaoctadecan-18-oic acid | PoSSuM | |||
FRZ | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-C]pyridazin-3-amine | PoSSuM | |||
GOL | Glycerol | PoSSuM |
Code | Name | Show |
---|---|---|
PTR | O-phosphotyrosine | |
TPO | Phosphothreonine |
Code | Name | Emphasize |
---|
Code | Name | Show |
---|
Download interaction data: 5V61
Structure summary
Code : | 5V61 PDBj RCSB PDB PDBe | ||||||||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Header : | TRANSFERASE/INHIBITOR | ||||||||||||||||||||||||
Title : | Phospho-ERK2 bound to bivalent inhibitor SBP2 | ||||||||||||||||||||||||
Release Data : | 2017-07-26 | ||||||||||||||||||||||||
Compound : |
|
||||||||||||||||||||||||
Source : |
|
||||||||||||||||||||||||
Authors : | Lechtenberg, B.C., Riedl, S.J. | ||||||||||||||||||||||||
Keywords : | kinase, MAPK, phosphorylation, cancer, TRANSFERASE-TRANSFERASE INHIBITOR complex, TRANSFERASE-INHIBITOR complex | ||||||||||||||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.20 Å ) | ||||||||||||||||||||||||
Citation : |
Structure-Guided Strategy for the Development of Potent Bivalent ERK Inhibitors.
Lechtenberg, B.C.,Mace, P.D.,Sessions, E.H.
et al.
PubMed: 28740606 |
Reaction
Chain : | A | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
UniProt : | P28482 (MK01_HUMAN) | ||||||||||||
|
Chain : | I | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
UniProt : | Q15418 (KS6A1_HUMAN) | ||||||||||||
|
Chain : | I |
---|---|
UniProt : | P04608 (TAT_HV1H2) |
Reaction : | - |