PDB ID: 5QIM
Hetero Atom Contents
The number of atoms exceeds 100,000. So, it can not be displayed here.
Select unit:
Select hetatm:
Select chain: Sequence
Data format:
Color scheme of protein:
Structure summary
Code : | 5QIM PDBj RCSB PDB PDBe | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | TGF-BETA RECEPTOR TYPE 1 KINASE DOMAIN (T204D) IN COMPLEX WITH N-{4-[3-(5-METHOXYPYRIDIN-2-YL)-1H-PYRROLO[3,2-B] PYRIDIN-2-YL]PYRIDIN-2-YL}ACETAMIDE | ||||||||||||
Release Data : | 2018-10-31 | ||||||||||||
Compound : |
|
||||||||||||
Source : |
|
||||||||||||
Authors : | Sheriff, S. | ||||||||||||
Keywords : | ALK5, SB431542, KINASE DOMAIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX, TRANSFERASE | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.7500 Å ) | ||||||||||||
Citation : |
Discovery of 4-Azaindole Inhibitors of TGF beta RI as Immuno-oncology Agents.
Zhang, Y.,Zhao, Y.,Tebben, A.J.
et al.
PubMed: 30429955 |
Reaction
Chain : | A | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
UniProt : | P36897 (TGFR1_HUMAN) | ||||||||||||
|