Het-PDB Navi2 (PDB: 5O5A)

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Ligands
Code	Name		Style	Show	Link
9LN	1-ethyl-~{N}-methyl-2,3-bis(oxidanylidene)-~{N}-[(1-phenylpyrazol-4-yl)methyl]-4~{H}-quinoxaline-6-carboxamide				PoSSuM
NO3	Nitrate ion				PoSSuM

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Download interaction data: 5O5A

Code :

5O5A PDBj RCSB PDB PDBe

Header :

DNA BINDING PROTEIN

Title :

Crystal structure of the human BRPF1 bromodomain in complex with BZ032

Release Data :

2018-06-13

Compound :

mol_id	molecule	chains	synonym
1	Peregrin	A	Bromodomain and PHD finger-containing protein 1,Protein Br140

Source :

mol_id	organism_scientific	organism_common	expression_system
1	Homo sapiens (taxid:9606)	Human	Escherichia coli (taxid:562)
	gene: BRPF1, BR140

Authors :

Zhu, J., Caflisch, A.

Keywords :

Bromodomain and PHD finger-containing protein 1(BRPF1), monocytic leukemia zinc-finger (MOZ), Inhibitor, transcription, DNA binding protein

Exp. method :

X-RAY DIFFRACTION ( 1.600 Å )

Citation :

Structure-based discovery of selective BRPF1 bromodomain inhibitors.

Zhu, J.,Zhou, C.,Caflisch, A.
(2018) Eur J Med Chem 155 : 337 - 352

PDB ID: 5O5A