PDB ID: 5O3G
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Code | Name | Style | Show | Link | |
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9J8 | (2~{R})-2-[(4~{S})-6-(4-chlorophenyl)-8-methoxy-1-methyl-4~{H}-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-~{N}-ethyl-pent-4-enamide | PoSSuM |
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Download interaction data: 5O3G
Structure summary
Code : | 5O3G PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSCRIPTION | ||||||||||||
Title : | Human Brd2(BD2) mutant in complex with AL-Am1 | ||||||||||||
Release Data : | 2018-02-14 | ||||||||||||
Compound : |
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Authors : | Chan, K.-H., Runcie, A.C., Ciulli, A. | ||||||||||||
Keywords : | The Bromodomain and Extra-Terminal Domain (BET) Family Chromatin binding protein, transcription | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.850 Å ) | ||||||||||||
Citation : |
Optimization of a "bump-and-hole" approach to allele-selective BET bromodomain inhibition.
Runcie, A.C.,Zengerle, M.,Chan, K.H.
et al.
PubMed: 29732121 |
Reaction
Chain : | A, B |
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UniProt : | P25440 (BRD2_HUMAN) |
Reaction : | - |