PDB ID: 5NU5
Hetero Atom Contents
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Code | Name | Style | Show | Link | |
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99E | ~{N}-[[2,8-bis(oxidanyl)naphthalen-1-yl]methyl]-4-ethanoyl-3-ethyl-5-methyl-1~{H}-pyrrole-2-carboxamide | PoSSuM | |||
EDO | 1,2-ethanediol | PoSSuM |
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Download interaction data: 5NU5
Structure summary
Code : | 5NU5 PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE | ||||||||||||
Title : | Crystal structure of the human bromodomain of EP300 bound to the inhibitor XDM-CBP | ||||||||||||
Release Data : | 2017-08-16 | ||||||||||||
Compound : |
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Authors : | Huegle, M., Wohlwend, D. | ||||||||||||
Keywords : | bromodomain, protein-inhibitor complex, epigenetics, EP300, transferase | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.6000 Å ) | ||||||||||||
Citation : |
Beyond the BET Family: Targeting CBP/p300 with 4-Acyl Pyrroles.
Hugle, M.,Lucas, X.,Ostrovskyi, D.
et al.
PubMed: 28766825 |
Reaction
Chain : | A, B | |||||||||||||||||||||||||||||
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UniProt : | Q09472 (EP300_HUMAN) | |||||||||||||||||||||||||||||
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