PDB ID: 5AL5
Hetero Atom Contents
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Color scheme of protein:
Code | Name | Style | Show | Link | |
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ZN | Zinc ion | PoSSuM | |||
SO4 | Sulfate ion | PoSSuM | |||
JL9 | 2-(4-((pyridin-4-yl)methyl)piperazin-1-yl)-3,4,5,6,7,8-hexahydroquinazolin-4-one | PoSSuM | |||
GOL | Glycerol | PoSSuM |
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Download interaction data: 5AL5
Structure summary
Code : | 5AL5 PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE | ||||||||||||
Title : | Crystal structure of TNKS2 in complex with 2-(4-((pyridin-4-yl)methyl) piperazin-1-yl)-3,4,5,6,7,8-hexahydroquinazolin-4-one | ||||||||||||
Release Data : | 2015-07-29 | ||||||||||||
Compound : |
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Source : |
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Authors : | Nkizinkiko, Y., Lehtio, L. | ||||||||||||
Keywords : | TRANSFERASE, PROTEIN-LIGAND COMPLEX, DIPHTHERIA TOXIN LIKE FOLD, ADP- RIBOSYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.05 Å ) | ||||||||||||
Citation : |
Discovery of Potent and Selective Nonplanar Tankyrase Inhibiting Nicotinamide Mimics.
Nkizinkiko, Y.,Suneel Kumar, B.V.S.,Jeankumar, V.U.
et al.
PubMed: 26183543 |
Reaction
Chain : | A, B | ||||||||||||||||
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UniProt : | Q9H2K2 (TNKS2_HUMAN) | ||||||||||||||||
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