PDB ID: 4ZHX
Hetero Atom Contents
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Color scheme of protein:
Code | Name | Style | Show | Link | |
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4O7 | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,1 5-triazadibenzo[B,H]cyclonona[1,2,3,4-jkl]cyclopenta[E]-as-indacen-14-ol | PoSSuM | |||
C1V | 3-[4-(2-hydroxyphenyl)phenyl]-4-oxidanyl-6-oxidanylidene-7h-thieno[2,3-B]pyridine-5-carbonitrile | PoSSuM | |||
C2Z | 5-(5-hydroxyl-isoxazol-3-yl)-furan-2-phosphonic acid | PoSSuM |
Code | Name | Show |
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TPO | Phosphothreonine | |
SEP | Phosphoserine |
Code | Name | Emphasize |
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Code | Name | Show |
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Download interaction data: 4ZHX
Structure summary
Code : | 4ZHX PDBj RCSB PDB PDBe | ||||||||||||||||||||||||||||||||||||
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Header : | TRANSFERASE | ||||||||||||||||||||||||||||||||||||
Title : | Novel binding site for allosteric activation of AMPK | ||||||||||||||||||||||||||||||||||||
Release Data : | 2016-03-09 | ||||||||||||||||||||||||||||||||||||
Compound : |
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Source : |
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Authors : | Langendorf, C.G., Ngoei, K.R., Issa, S.M.A., Ling, N., Gorman, M.A., Parker, M.W., Sakamoto, K., Scott, J.W., Oakhill, J.S., Kemp, B.E. | ||||||||||||||||||||||||||||||||||||
Keywords : | Transferase, serine/threonine kinase, allosteric activation, nucleotide-binding | ||||||||||||||||||||||||||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.9900 Å ) | ||||||||||||||||||||||||||||||||||||
Citation : |
Structural basis of allosteric and synergistic activation of AMPK by furan-2-phosphonic derivative C2 binding.
Langendorf, C.G.,Ngoei, K.R.,Scott, J.W.
et al.
PubMed: 26952388 |
Reaction
Chain : | A, C | ||||||||||||||||||||
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UniProt : | P54646 (AAPK2_HUMAN) | ||||||||||||||||||||
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Chain : | B, D |
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UniProt : | Q9Y478 (AAKB1_HUMAN) |
Reaction : | - |
Chain : | E, F |
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UniProt : | P54619 (AAKG1_HUMAN) |
Reaction : | - |