PDB ID: 4UYE
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Structure summary
Code : | 4UYE PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSCRIPTION | ||||||||||||
Title : | BROMODOMAIN OF HUMAN BRPF1 WITH N-1,3-dimethyl-2-oxo-6-(piperidin-1- yl)-2,3-dihydro-1H-1,3-benzodiazol-5-yl-2-methoxybenzamide | ||||||||||||
Release Data : | 2014-09-17 | ||||||||||||
Compound : |
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Source : |
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Authors : | Chung, C., Bamborough, P., Demont, E. | ||||||||||||
Keywords : | TRANSCRIPTION, INHIBITOR, HISTONE, EPIGENETIC READER, ANTAGONIST | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.65 Å ) | ||||||||||||
Citation : |
1,3-Dimethyl Benzimidazolones are Potent, Selective Inhibitors of the Brpf1 Bromodomain.
Demont, E.H.,Bamborough, P.,Chung, C.W.
et al.
PubMed: 25408830 |
Reaction
Chain : | A, B |
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UniProt : | P55201 (BRPF1_HUMAN) |
Reaction : | - |