PDB ID: 4E47
Hetero Atom Contents
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Code | Name | Style | Show | Link | |
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SAM | S-adenosylmethionine | PoSSuM | |||
0N6 | (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide | PoSSuM | |||
BME | Beta-mercaptoethanol | PoSSuM | |||
SO4 | Sulfate ion | PoSSuM |
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Download interaction data: 4E47
Structure summary
Code : | 4E47 PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | SET7/9 in complex with inhibitor (R)-(3-(3-cyanophenyl)-1-oxo-1-(pyrrolidin-1-yl)propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-6- sulfonamide and S-adenosylmethionine | ||||||||||||
Release Data : | 2012-03-28 | ||||||||||||
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Authors : | Walker, J.R., Ouyang, H., Dong, A., Fish, P., Cook, A., Barsyte, D., Vedadi, M., Tatlock, J., Owen, D., Bunnage, M., Bountra, C., Weigelt, J., Edwards, A.M., Arrowsmith, C.H., Brown, P.J., Structural Genomics Consortium (SGC) | ||||||||||||
Keywords : | ternary complex, SET domain, methyltransferase, inhibitor, S-adenosylmethionine, chromatin regulator, chromosomal protein, nucleus, transcription, transcription regulation, transferase, Structural Genomics Consortium, SGC, TRANSFERASE-TRANSFERASE INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.00 Å ) | ||||||||||||
Citation : |
Setd7 in Complex with Inhibitor and SAM
Walker, J.R.,Ouyang, H.,Dong, A.
et al.
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Reaction
Chain : | A, B, C, D | ||||||||||||
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UniProt : | Q8WTS6 (SETD7_HUMAN) | ||||||||||||
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