PDB ID: 4BVF
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Structure summary
Code : | 4BVF PDBj RCSB PDB PDBe | ||||||||||||||||||||||||
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Header : | HYDROLASE/LIGASE | ||||||||||||||||||||||||
Title : | CRYSTAL STRUCTURE OF HUMAN SIRT3 IN COMPLEX WITH THIOALKYLIMIDATE FORMED FROM THIO-ACETYL-LYSINE ACS2-PEPTIDE CRYSTALLIZED IN PRESENCE OF THE INHIBITOR EX-527 | ||||||||||||||||||||||||
Release Data : | 2013-07-17 | ||||||||||||||||||||||||
Compound : |
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Source : |
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Authors : | Gertz, M., Weyand, M., Steegborn, C. | ||||||||||||||||||||||||
Keywords : | HYDROLASE-LIGASE COMPLEX, THIO-INTERMEDIATE, HYDROLASE-HYDROLASE | ||||||||||||||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.70 Å ) | ||||||||||||||||||||||||
Citation : |
Ex-527 Inhibits Sirtuins by Exploiting Their Unique Nad+-Dependent Deacetylation Mechanism
Gertz, M.,Fischer, F.,Nguyen, G.T.T.
et al.
PubMed: 23840057 |
Reaction
Chain : | A | ||||||||
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UniProt : | Q9NTG7 (SIR3_HUMAN) | ||||||||
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Chain : | B | ||||||||||||
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UniProt : | Q9NUB1 (ACS2L_HUMAN) | ||||||||||||
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