PDB ID: 3V8S
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Structure summary
Code : | 3V8S PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | Human RHO-ASSOCIATED PROTEIN KINASE 1 (ROCK 1) IN COMPLEX WITH INDAZOLE DERIVATIVE (COMPOUND 18) | ||||||||||||
Release Data : | 2012-02-08 | ||||||||||||
Compound : |
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Source : |
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Authors : | Martin, M.P., Zhu, J.-Yi., Schonbrunn, E. | ||||||||||||
Keywords : | KINASE, DIMERIZATION, MYOSIN, TRANSFERASE, INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.286 Å ) | ||||||||||||
Citation : |
Fragment-based and structure-guided discovery and optimization of rho kinase inhibitors.
Li, R.,Martin, M.P.,Liu, Y.
et al.
PubMed: 22272748 |
Reaction
Chain : | A, B, C, D | |||||||||||||
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UniProt : | Q13464 (ROCK1_HUMAN) | |||||||||||||
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