PDB ID: 3PVU
Hetero Atom Contents
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Code | Name | Style | Show | Link | |
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QRW | 3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-N-[2-(trifluoromethyl)benzyl]benzamide | PoSSuM |
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CMT | O-methylcysteine |
Code | Name | Emphasize |
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Download interaction data: 3PVU
Structure summary
Code : | 3PVU PDBj RCSB PDB PDBe | ||||||||||||||||||||||||||||||||||||
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Header : | TRANSFERASE/SIGNALING PROTEIN/INHIBITOR | ||||||||||||||||||||||||||||||||||||
Title : | Bovine GRK2 in complex with Gbetagamma subunits and a selective kinase inhibitor (CMPD101) | ||||||||||||||||||||||||||||||||||||
Release Data : | 2011-06-01 | ||||||||||||||||||||||||||||||||||||
Compound : |
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Source : |
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Authors : | Thal, D.M., Tesmer, J.J. | ||||||||||||||||||||||||||||||||||||
Keywords : | Transferase, Serine/threonine-protein kinase, ATP-binding, Inhibitor, Membrane, TRANSFERASE-SIGNALING PROTEIN-INHIBITOR complex | ||||||||||||||||||||||||||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.4800 Å ) | ||||||||||||||||||||||||||||||||||||
Citation : |
Molecular Mechanism of Selectivity among G Protein-Coupled Receptor Kinase 2 Inhibitors.
Thal, D.M.,Yeow, R.Y.,Schoenau, C.
et al.
PubMed: 21596927 |
Reaction
Chain : | A | ||||||||
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UniProt : | P21146 (ARBK1_BOVIN) | ||||||||
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Chain : | B |
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UniProt : | P62871 (GBB1_BOVIN) |
Reaction : | - |
Chain : | G |
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UniProt : | P63212 (GBG2_BOVIN) |
Reaction : | - |