PDB ID: 3UVQ
Hetero Atom Contents
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FS8 | N-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,D][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | PoSSuM | |||
BOG | Octyl beta-D-glucopyranoside | PoSSuM |
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Download interaction data: 3UVQ
Structure summary
Code : | 3UVQ PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||
Title : | Human p38 MAP Kinase in Complex with a Dibenzosuberone Derivative | ||||||||||||
Release Data : | 2012-12-05 | ||||||||||||
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Authors : | Mayer-Wrangowski, S.C., Richters, A., Gruetter, C., Rauh, D. | ||||||||||||
Keywords : | selective p38 inhibitor, SAR, dibenzosuberone derivative, protein kinase, TRANSFERASE-TRANSFERASE INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.2000 Å ) | ||||||||||||
Citation : |
Dibenzosuberones as p38 mitogen-activated protein kinase inhibitors with low ATP competitiveness and outstanding whole blood activity.
Fischer, S.,Wentsch, H.K.,Mayer-Wrangowski, S.C.
et al.
PubMed: 23270382 |
Reaction
Chain : | A | |||||||||||||
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UniProt : | Q16539 (MK14_HUMAN) | |||||||||||||
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