PDB ID: 3U5K
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Structure summary
Code : | 3U5K PDBj RCSB PDB PDBe | ||||||||||||
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Header : | SIGNALING PROTEIN/INHIBITOR | ||||||||||||
Title : | Crystal Structure of the first bromodomain of human BRD4 in complex with Midazolam | ||||||||||||
Release Data : | 2011-11-23 | ||||||||||||
Compound : |
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Source : |
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Authors : | Filippakopoulos, P., Picaud, S., Felletar, I., Fedorov, O., von Delft, F., Arrowsmith, C.H., Edwards, A.M., Weigelt, J., Bountra, C., Knapp, S., Structural Genomics Consortium (SGC) | ||||||||||||
Keywords : | Bromodomain-containing protein 4 isoform long, BRD4, Bromodomain containing protein 4, CAP, HUNK1, MCAP, Mitotic chromosome associated protein, Structural Genomics Consortium, SGC, SIGNALING PROTEIN-INHIBITOR complex | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.8000 Å ) | ||||||||||||
Citation : |
Benzodiazepines and benzotriazepines as protein interaction inhibitors targeting bromodomains of the BET family.
Filippakopoulos, P.,Picaud, S.,Fedorov, O.
et al.
PubMed: 22137933 |
Reaction
Chain : | A, B, C, D |
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UniProt : | O60885 (BRD4_HUMAN) |
Reaction : | - |