PDB ID: 2XCH
Hetero Atom Contents
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Color scheme of protein:
Code | Name | Style | Show | Link | |
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CKG | 8-(cyclohexa-2,5-dien-1-ylideneamino)-1-(piperidin-4-ylmethyl)-4,5-dihydro-1h-pyrazolo[4,3-H]quinazoline-3-carboxamide | PoSSuM | |||
GOL | Glycerol | PoSSuM | |||
SO4 | Sulfate ion | PoSSuM |
Code | Name | Show |
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SEP | Phosphoserine |
Code | Name | Emphasize |
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Code | Name | Show |
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Download interaction data: 2XCH
Structure summary
Code : | 2XCH PDBj RCSB PDB PDBe | ||||||||||||
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Header : | TRANSFERASE | ||||||||||||
Title : | Crystal structure of PDK1 in complex with a pyrazoloquinazoline inhibitor | ||||||||||||
Release Data : | 2010-07-28 | ||||||||||||
Compound : |
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Source : |
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Authors : | Angiolini, M., Banfi, P., Casale, E., Casuscelli, F., Fiorelli, C., Saccardo, M.B., Silvagni, M., Zuccotto, F. | ||||||||||||
Keywords : | PI3-KINASE SIGNALLING, TRANSFERASE, SERINE/THREONINE-PROTEIN KINASE, ATP-BINDING | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.00 Å ) | ||||||||||||
Citation : |
Structure-Based Optimization of Potent Pdk1 Inhibitors.
Angiolini, M.,Banfi, P.,Casale, E.
et al.
PubMed: 20621725 |
Reaction
Chain : | A | ||||||||||||
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UniProt : | O15530 (PDPK1_HUMAN) | ||||||||||||
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