PDB ID: 2VQM
Hetero Atom Contents
The number of atoms exceeds 100,000. So, it can not be displayed here.
Select unit:
Select hetatm:
Select chain: Sequence
Data format:
Color scheme of protein:
Code | Name | Style | Show | Link | |
---|---|---|---|---|---|
HA3 | N-hydroxy-5-[(3-phenyl-5,6-dihydroimidazo[1,2-a]pyrazin-7(8h)-yl)carbonyl]thiophene-2-carboxamide | PoSSuM | |||
K | Potassium ion | PoSSuM | |||
ZN | Zinc ion | PoSSuM |
Code | Name | Show |
---|
Code | Name | Emphasize |
---|
Code | Name | Show |
---|
Download interaction data: 2VQM
Structure summary
Code : | 2VQM PDBj RCSB PDB PDBe | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Header : | HYDROLASE | ||||||||||||
Title : | Structure of HDAC4 catalytic domain bound to a hydroxamic acid inhbitor | ||||||||||||
Release Data : | 2008-07-08 | ||||||||||||
Compound : |
|
||||||||||||
Source : |
|
||||||||||||
Authors : | Bottomley, M.J., Lo Surdo, P., Di Giovine, P., Cirillo, A., Scarpelli, R., Ferrigno, F., Jones, P., Neddermann, P., De Francesco, R., Steinkuhler, C., Gallinari, P., Carfi, A. | ||||||||||||
Keywords : | INHIBITOR, REPRESSOR, CHROMATIN, COILED COIL, HISTONE DEACETYLASE, TRANSCRIPTION REGULATION, UBL CONJUGATION, CHROMATIN REGULATOR, POLYMORPHISM, TRANSCRIPTION, PHOSPHOPROTEIN, HDAC, ZINC, HDACI, NUCLEUS, HYDROLASE, CYTOPLASM | ||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 1.80 Å ) | ||||||||||||
Citation : |
Structural and Functional Analysis of the Human Hdac4 Catalytic Domain Reveals a Regulatory Zinc-Binding Domain.
Bottomley, M.J.,Lo Surdo, P.,Di Giovine, P.
et al.
PubMed: 18614528 |
Reaction
Chain : | A | |||||||||
---|---|---|---|---|---|---|---|---|---|---|
UniProt : | P56524 (HDAC4_HUMAN) | |||||||||
|