PDB ID: 1JCR
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Structure summary
Code : | 1JCR PDBj RCSB PDB PDBe | ||||||||||||||||||||||||||||||||||||
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Header : | TRANSFERASE/TRANSFERASE INHIBITOR | ||||||||||||||||||||||||||||||||||||
Title : | CRYSTAL STRUCTURE OF RAT PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH THE NON-SUBSTRATE TETRAPEPTIDE INHIBITOR CVFM AND FARNESYL DIPHOSPHATE SUBSTRATE | ||||||||||||||||||||||||||||||||||||
Release Data : | 2001-11-02 | ||||||||||||||||||||||||||||||||||||
Compound : |
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Source : |
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Authors : | Long, S.B., Casey, P.J., Beese, L.S. | ||||||||||||||||||||||||||||||||||||
Keywords : | FTASE, PFT, PFTASE, FT, FPT, FARNESYLTRANSFERASE, FARNESYL TRANSFERASE, FARNESYL PROTEIN TRANSFERASE, CAAX, RAS, CANCER, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX | ||||||||||||||||||||||||||||||||||||
Exp. method : | X-RAY DIFFRACTION ( 2.00 Å ) | ||||||||||||||||||||||||||||||||||||
Citation : |
The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics.
Long, S.B.,Hancock, P.J.,Kral, A.M.
et al.
PubMed: 11687658 The Basis for K-Ras4B Binding Specificity to Protein Farnesyltransferase Revealed by 2A Resolution Ternary Complex Structures
Long, S.B.,Casey, P.J.,Beese, L.S.
Crystal Structure of Protein Farnesyltransferase at 2.25A Resolution
Park, H.-W.,Boduluri, S.R.,Moomaw, J.F.
et al.
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Reaction
Chain : | A | ||||||||||||
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UniProt : | Q04631 (FNTA_RAT) | ||||||||||||
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Chain : | B | ||||||||
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UniProt : | Q02293 (FNTB_RAT) | ||||||||
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