ID 5VALA STANDARD; PRT; 281 AA. DT CONVERTED FROM PDB (SEQRES) 5VAL DE Serine/threonine-protein kinase B-raf OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.260 CC R-Factor 0.183 FT #SUB 4 446 SER A 64 506 ARG B Protein B 9 FT #SUB 5 447 SER A 64 506 ARG B Protein B 3 FT #SUB 5 447 SER A 65 507 LYS B Protein B 4 FT #SUB 6 448 ASP A 8 450 TRP B Protein S 7 FT #SUB 6 448 ASP A 64 506 ARG B Protein A 10 FT #SUB 6 448 ASP A 65 507 LYS B Protein B 1 FT #SUB 6 448 ASP A 67 509 ARG B Protein A 6 FT #SUB 7 449 ASP A 67 509 ARG B Protein B 2 FT #SUB 7 449 ASP A 128 570 LYS B Protein A 2 FT #SUB 8 450 TRP A 7 449 ASP B Protein S 2 FT #SUB 8 450 TRP A 67 509 ARG B Protein A 7 FT #SUB 34 476 TRP A 124 566 TYR B Protein S 2 FT #SUB 35 477 HIS A 68 510 HIS B Protein A 6 FT #SUB 35 477 HIS A 120 562 GLN B Protein B 6 FT #SUB 35 477 HIS A 123 565 ASP B Protein S 4 FT #SUB 35 477 HIS A 124 566 TYR B Protein S 3 FT #SUB 35 477 HIS A 127 569 ALA B Protein S 2 FT #SUB 36 478 GLY A 120 562 GLN B Protein B 5 FT #SUB 64 506 ARG A 8 450 TRP B Protein B 2 FT #SUB 65 507 LYS A 7 449 ASP B Protein S 2 FT #SUB 65 507 LYS A 8 450 TRP B Protein B 5 FT #SUB 66 508 THR A 8 450 TRP B Protein B 1 FT #SUB 67 509 ARG A 8 450 TRP B Protein S 14 FT #SUB 67 509 ARG A 63 505 LEU B Protein S 1 FT #SUB 67 509 ARG A 64 506 ARG B Protein S 4 FT #SUB 67 509 ARG A 66 508 THR B Protein S 5 FT #SUB 67 509 ARG A 67 509 ARG B Protein S 3 FT #SUB 67 509 ARG A 73 515 LEU B Protein B 1 FT #SUB 67 509 ARG A 74 516 PHE B Protein S 11 FT #SUB 67 509 ARG A 75 517 MET B Protein B 3 FT #SUB 68 510 HIS A 35 477 HIS B Protein S 6 FT #SUB 68 510 HIS A 73 515 LEU B Protein B 3 FT #SUB 68 510 HIS A 75 517 MET B Protein S 1 FT #SUB 69 511 VAL A 88 530 GLN B Protein S 2 FT #SUB 73 515 LEU A 67 509 ARG B Protein S 1 FT #SUB 73 515 LEU A 68 510 HIS B Protein S 3 FT #SUB 73 515 LEU A 73 515 LEU B Protein S 1 FT #SUB 74 516 PHE A 67 509 ARG B Protein B 3 FT #SUB 75 517 MET A 67 509 ARG B Protein A 7 FT #SUB 75 517 MET A 68 510 HIS B Protein S 1 FT #SUB 88 530 GLN A 69 511 VAL B Protein S 2 FT #SUB 120 562 GLN A 35 477 HIS B Protein S 6 FT #SUB 120 562 GLN A 36 478 GLY B Protein S 5 FT #SUB 123 565 ASP A 35 477 HIS B Protein A 4 FT #SUB 124 566 TYR A 35 477 HIS B Protein A 3 FT #SUB 127 569 ALA A 35 477 HIS B Protein S 2 FT #SUB 128 570 LYS A 7 449 ASP B Protein S 1 FT #SUB 128 570 LYS A 8 450 TRP B Protein S 2 FT #HET 21 463 ILE A 1 801 92D A S 2 FT #HET 29 471 VAL A 1 801 92D A S 3 FT #HET 39 481 ALA A 1 801 92D A A 7 FT #HET 40 482 VAL A 1 801 92D A B 2 FT #HET 41 483 LYS A 1 801 92D A A 4 FT #HET 59 501 GLU A 1 801 92D A S 10 FT #HET 62 504 VAL A 1 801 92D A S 1 FT #HET 63 505 LEU A 1 801 92D A S 3 FT #HET 72 514 LEU A 1 801 92D A S 6 FT #HET 85 527 ILE A 1 801 92D A A 2 FT #HET 87 529 THR A 1 801 92D A S 6 FT #HET 88 530 GLN A 1 801 92D A B 2 FT #HET 89 531 TRP A 1 801 92D A A 4 FT #HET 90 532 CYS A 1 801 92D A A 9 FT #HET 132 574 HIS A 1 801 92D A S 1 FT #HET 141 583 PHE A 1 801 92D A S 2 FT #HET 150 592 ILE A 1 801 92D A B 1 FT #HET 151 593 GLY A 1 801 92D A B 4 FT #HET 152 594 ASP A 1 801 92D A A 16 FT #HET 153 595 PHE A 1 801 92D A S 8 FT DISORDER 1 3 FT DISORDER 155 173 FT DISORDER 186 187 FT DISORDER 279 281 CC SEQUENCE 254 AA (ATOM); CC SSDDWEIPDG QITVGQRIGS GSFGTVYKGK WHGDVAVKML NVTAPTPQQL QAFKNEVGVL CC RKTRHVNILL FMGYSTKPQL AIVTQWCEGS SLYHHLHIIE TKFEMIKLID IARQTAQGMD CC YLHAKSIIHR DLKSNNIFLH EDLTVKIGDF GSILWMAPEV IRMKNPYSFQ SDVYAFGIVL CC YELMTGQLPY SNINNRDQII FMVGRGYLSP DLSKVRSNCP KAMKRLMAEC LKKKRDERPL CC FPQILASIEL LARS CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES GSDSSDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTP CC ATOM ---SSDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTP CC *********************************************** CC SEQRES QQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLH CC ATOM QQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLH CC ************************************************** CC SEQRES IIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKI CC ATOM IIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKI CC ************************************************** CC SEQRES GDFGLATVKSRWSGSHQFEQLSGSILWMAPEVIRMQDKNPYSFQSDVYAF CC ATOM GDFG-------------------SILWMAPEVIRM--KNPYSFQSDVYAF CC **** ************ ************* CC SEQRES GIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRL CC ATOM GIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRL CC ************************************************** CC SEQRES MAECLKKKRDERPLFPQILASIELLARSLPK CC ATOM MAECLKKKRDERPLFPQILASIELLARS--- CC **************************** SQ SEQUENCE 281 AA; MW; CN; GSDSSDDWEI PDGQITVGQR IGSGSFGTVY KGKWHGDVAV KMLNVTAPTP QQLQAFKNEV GVLRKTRHVN ILLFMGYSTK PQLAIVTQWC EGSSLYHHLH IIETKFEMIK LIDIARQTAQ GMDYLHAKSI IHRDLKSNNI FLHEDLTVKI GDFGLATVKS RWSGSHQFEQ LSGSILWMAP EVIRMQDKNP YSFQSDVYAF GIVLYELMTG QLPYSNINNR DQIIFMVGRG YLSPDLSKVR SNCPKAMKRL MAECLKKKRD ERPLFPQILA SIELLARSLP K // ID 5VALB STANDARD; PRT; 281 AA. DT CONVERTED FROM PDB (SEQRES) 5VAL DE Serine/threonine-protein kinase B-raf OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.260 CC R-Factor 0.183 FT #SUB 7 449 ASP B 8 450 TRP A Protein S 2 FT #SUB 7 449 ASP B 65 507 LYS A Protein S 2 FT #SUB 7 449 ASP B 128 570 LYS A Protein B 1 FT #SUB 8 450 TRP B 6 448 ASP A Protein S 7 FT #SUB 8 450 TRP B 64 506 ARG A Protein S 2 FT #SUB 8 450 TRP B 65 507 LYS A Protein S 5 FT #SUB 8 450 TRP B 66 508 THR A Protein S 1 FT #SUB 8 450 TRP B 67 509 ARG A Protein S 14 FT #SUB 8 450 TRP B 128 570 LYS A Protein S 2 FT #SUB 35 477 HIS B 68 510 HIS A Protein A 6 FT #SUB 35 477 HIS B 120 562 GLN A Protein B 6 FT #SUB 35 477 HIS B 123 565 ASP A Protein S 4 FT #SUB 35 477 HIS B 124 566 TYR A Protein S 3 FT #SUB 35 477 HIS B 127 569 ALA A Protein S 2 FT #SUB 36 478 GLY B 120 562 GLN A Protein B 5 FT #SUB 63 505 LEU B 67 509 ARG A Protein B 1 FT #SUB 64 506 ARG B 4 446 SER A Protein S 9 FT #SUB 64 506 ARG B 5 447 SER A Protein S 3 FT #SUB 64 506 ARG B 6 448 ASP A Protein A 10 FT #SUB 64 506 ARG B 67 509 ARG A Protein B 4 FT #SUB 65 507 LYS B 5 447 SER A Protein S 4 FT #SUB 65 507 LYS B 6 448 ASP A Protein B 1 FT #SUB 66 508 THR B 67 509 ARG A Protein B 5 FT #SUB 67 509 ARG B 6 448 ASP A Protein S 6 FT #SUB 67 509 ARG B 7 449 ASP A Protein S 2 FT #SUB 67 509 ARG B 8 450 TRP A Protein S 7 FT #SUB 67 509 ARG B 67 509 ARG A Protein S 3 FT #SUB 67 509 ARG B 73 515 LEU A Protein B 1 FT #SUB 67 509 ARG B 74 516 PHE A Protein S 3 FT #SUB 67 509 ARG B 75 517 MET A Protein A 7 FT #SUB 68 510 HIS B 35 477 HIS A Protein S 6 FT #SUB 68 510 HIS B 73 515 LEU A Protein B 3 FT #SUB 68 510 HIS B 75 517 MET A Protein S 1 FT #SUB 69 511 VAL B 88 530 GLN A Protein S 2 FT #SUB 73 515 LEU B 67 509 ARG A Protein S 1 FT #SUB 73 515 LEU B 68 510 HIS A Protein S 3 FT #SUB 73 515 LEU B 73 515 LEU A Protein S 1 FT #SUB 74 516 PHE B 67 509 ARG A Protein A 11 FT #SUB 75 517 MET B 67 509 ARG A Protein S 3 FT #SUB 75 517 MET B 68 510 HIS A Protein S 1 FT #SUB 88 530 GLN B 69 511 VAL A Protein S 2 FT #SUB 120 562 GLN B 35 477 HIS A Protein S 6 FT #SUB 120 562 GLN B 36 478 GLY A Protein S 5 FT #SUB 123 565 ASP B 35 477 HIS A Protein A 4 FT #SUB 124 566 TYR B 34 476 TRP A Protein S 2 FT #SUB 124 566 TYR B 35 477 HIS A Protein A 3 FT #SUB 127 569 ALA B 35 477 HIS A Protein S 2 FT #SUB 128 570 LYS B 7 449 ASP A Protein S 2 FT #HET 21 463 ILE B 2 801 92D B S 1 FT #HET 29 471 VAL B 2 801 92D B S 3 FT #HET 39 481 ALA B 2 801 92D B A 7 FT #HET 40 482 VAL B 2 801 92D B B 2 FT #HET 41 483 LYS B 2 801 92D B A 5 FT #HET 59 501 GLU B 2 801 92D B S 9 FT #HET 63 505 LEU B 2 801 92D B S 3 FT #HET 72 514 LEU B 2 801 92D B S 6 FT #HET 85 527 ILE B 2 801 92D B A 2 FT #HET 87 529 THR B 2 801 92D B S 6 FT #HET 88 530 GLN B 2 801 92D B B 2 FT #HET 89 531 TRP B 2 801 92D B A 3 FT #HET 90 532 CYS B 2 801 92D B A 9 FT #HET 130 572 ILE B 2 801 92D B S 1 FT #HET 132 574 HIS B 2 801 92D B S 1 FT #HET 141 583 PHE B 2 801 92D B S 1 FT #HET 151 593 GLY B 2 801 92D B B 4 FT #HET 152 594 ASP B 2 801 92D B A 14 FT #HET 153 595 PHE B 2 801 92D B S 8 FT DISORDER 1 5 FT DISORDER 156 172 FT DISORDER 186 188 FT DISORDER 280 281 CC SEQUENCE 254 AA (ATOM); CC DDWEIPDGQI TVGQRIGSGS FGTVYKGKWH GDVAVKMLNV TAPTPQQLQA FKNEVGVLRK CC TRHVNILLFM GYSTKPQLAI VTQWCEGSSL YHHLHIIETK FEMIKLIDIA RQTAQGMDYL CC HAKSIIHRDL KSNNIFLHED LTVKIGDFGL GSILWMAPEV IRMNPYSFQS DVYAFGIVLY CC ELMTGQLPYS NINNRDQIIF MVGRGYLSPD LSKVRSNCPK AMKRLMAECL KKKRDERPLF CC PQILASIELL ARSL CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES GSDSSDDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTP CC ATOM -----DDWEIPDGQITVGQRIGSGSFGTVYKGKWHGDVAVKMLNVTAPTP CC ********************************************* CC SEQRES QQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLH CC ATOM QQLQAFKNEVGVLRKTRHVNILLFMGYSTKPQLAIVTQWCEGSSLYHHLH CC ************************************************** CC SEQRES IIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKI CC ATOM IIETKFEMIKLIDIARQTAQGMDYLHAKSIIHRDLKSNNIFLHEDLTVKI CC ************************************************** CC SEQRES GDFGLATVKSRWSGSHQFEQLSGSILWMAPEVIRMQDKNPYSFQSDVYAF CC ATOM GDFGL-----------------GSILWMAPEVIRM---NPYSFQSDVYAF CC ***** ************* ************ CC SEQRES GIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRL CC ATOM GIVLYELMTGQLPYSNINNRDQIIFMVGRGYLSPDLSKVRSNCPKAMKRL CC ************************************************** CC SEQRES MAECLKKKRDERPLFPQILASIELLARSLPK CC ATOM MAECLKKKRDERPLFPQILASIELLARSL-- CC ***************************** SQ SEQUENCE 281 AA; MW; CN; GSDSSDDWEI PDGQITVGQR IGSGSFGTVY KGKWHGDVAV KMLNVTAPTP QQLQAFKNEV GVLRKTRHVN ILLFMGYSTK PQLAIVTQWC EGSSLYHHLH IIETKFEMIK LIDIARQTAQ GMDYLHAKSI IHRDLKSNNI FLHEDLTVKI GDFGLATVKS RWSGSHQFEQ LSGSILWMAP EVIRMQDKNP YSFQSDVYAF GIVLYELMTG QLPYSNINNR DQIIFMVGRG YLSPDLSKVR SNCPKAMKRL MAECLKKKRD ERPLFPQILA SIELLARSLP K //