ID 4G9CA STANDARD; PRT; 307 AA. DT CONVERTED FROM PDB (SEQRES) 4G9C DE Serine/threonine-protein kinase B-raf OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 3.500 CC R-Factor 0.262 FT #SUB 29 448 ASP A 87 506 ARG B Protein S 6 FT #SUB 29 448 ASP A 88 507 LYS B Protein S 1 FT #SUB 31 450 TRP A 87 506 ARG B Protein S 2 FT #SUB 31 450 TRP A 88 507 LYS B Protein S 2 FT #SUB 31 450 TRP A 90 509 ARG B Protein S 7 FT #SUB 57 476 TRP A 147 566 TYR B Protein S 1 FT #SUB 58 477 HIS A 91 510 HIS B Protein B 2 FT #SUB 58 477 HIS A 143 562 GLN B Protein B 4 FT #SUB 58 477 HIS A 146 565 ASP B Protein S 3 FT #SUB 58 477 HIS A 150 569 ALA B Protein S 2 FT #SUB 59 478 GLY A 143 562 GLN B Protein B 5 FT #SUB 86 505 LEU A 90 509 ARG B Protein B 1 FT #SUB 87 506 ARG A 29 448 ASP B Protein A 8 FT #SUB 87 506 ARG A 31 450 TRP B Protein B 2 FT #SUB 87 506 ARG A 90 509 ARG B Protein B 1 FT #SUB 88 507 LYS A 29 448 ASP B Protein S 1 FT #SUB 88 507 LYS A 31 450 TRP B Protein B 3 FT #SUB 89 508 THR A 90 509 ARG B Protein B 3 FT #SUB 90 509 ARG A 31 450 TRP B Protein S 9 FT #SUB 90 509 ARG A 86 505 LEU B Protein S 1 FT #SUB 90 509 ARG A 87 506 ARG B Protein S 1 FT #SUB 90 509 ARG A 89 508 THR B Protein S 3 FT #SUB 90 509 ARG A 90 509 ARG B Protein S 8 FT #SUB 90 509 ARG A 96 515 LEU B Protein S 2 FT #SUB 90 509 ARG A 97 516 PHE B Protein S 8 FT #SUB 90 509 ARG A 98 517 MET B Protein B 3 FT #SUB 91 510 HIS A 58 477 HIS B Protein S 6 FT #SUB 91 510 HIS A 96 515 LEU B Protein B 2 FT #SUB 91 510 HIS A 98 517 MET B Protein S 1 FT #SUB 96 515 LEU A 90 509 ARG B Protein S 3 FT #SUB 96 515 LEU A 91 510 HIS B Protein S 1 FT #SUB 97 516 PHE A 90 509 ARG B Protein A 12 FT #SUB 98 517 MET A 90 509 ARG B Protein S 1 FT #SUB 143 562 GLN A 58 477 HIS B Protein S 8 FT #SUB 143 562 GLN A 59 478 GLY B Protein S 7 FT #SUB 146 565 ASP A 58 477 HIS B Protein A 7 FT #SUB 147 566 TYR A 31 450 TRP B Protein S 1 FT #SUB 147 566 TYR A 57 476 TRP B Protein S 2 FT #SUB 147 566 TYR A 58 477 HIS B Protein A 4 FT #SUB 150 569 ALA A 58 477 HIS B Protein S 2 FT #SUB 151 570 LYS A 30 449 ASP B Protein S 1 FT #SUB 167 586 GLU A 169 588 LEU B Protein S 1 FT #SUB 169 588 LEU A 167 586 GLU B Protein S 1 FT #SUB 296 715 GLU A 56 475 LYS B Protein S 1 FT #HET 44 463 ILE A 1 801 0WP A S 3 FT #HET 52 471 VAL A 1 801 0WP A S 1 FT #HET 62 481 ALA A 1 801 0WP A A 6 FT #HET 63 482 VAL A 1 801 0WP A B 1 FT #HET 64 483 LYS A 1 801 0WP A A 4 FT #HET 82 501 GLU A 1 801 0WP A S 10 FT #HET 85 504 VAL A 1 801 0WP A S 1 FT #HET 86 505 LEU A 1 801 0WP A S 5 FT #HET 94 513 ILE A 1 801 0WP A S 1 FT #HET 95 514 LEU A 1 801 0WP A S 4 FT #HET 108 527 ILE A 1 801 0WP A A 6 FT #HET 110 529 THR A 1 801 0WP A S 11 FT #HET 111 530 GLN A 1 801 0WP A B 2 FT #HET 112 531 TRP A 1 801 0WP A A 15 FT #HET 113 532 CYS A 1 801 0WP A A 4 FT #HET 153 572 ILE A 1 801 0WP A S 1 FT #HET 155 574 HIS A 1 801 0WP A S 2 FT #HET 164 583 PHE A 1 801 0WP A S 4 FT #HET 174 593 GLY A 1 801 0WP A B 3 FT #HET 175 594 ASP A 1 801 0WP A A 14 FT #HET 176 595 PHE A 1 801 0WP A A 12 FT #HET 179 598 ALA A 1 801 0WP A S 1 FT #HET 180 599 THR A 1 801 0WP A B 1 FT DISORDER 1 28 FT DISORDER 183 193 FT DISORDER 305 307 CC SEQUENCE 265 AA (ATOM); CC DDWEIPDGQI TVGQRIGSGS FGTVYKGKWH GDVAVKMLNV TAPTPQQLQA FKNEVGVLRK CC TRHVNILLFM GYSTKPQLAI VTQWCEGSSL YHHLHIIETK FEMIKLIDIA RQTAQGMDYL CC HAKSIIHRDL KSNNIFLHED LTVKIGDFGL ATVKLSGSIL WMAPEVIRMQ DKNPYSFQSD CC VYAFGIVLYE LMTGQLPYSN INNRDQIIFM VGRGYLSPDL SKVRSNCPKA MKRLMAECLK CC KKRDERPLFP QILASIELLA RSLPK CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES MDRGSHHHHHHGSEDRNRMKTLGRRDSSDDWEIPDGQITVGQRIGSGSFG CC ATOM ----------------------------DDWEIPDGQITVGQRIGSGSFG CC ********************** CC SEQRES TVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGY CC ATOM TVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGY CC ************************************************** CC SEQRES STKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHA CC ATOM STKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHA CC ************************************************** CC SEQRES KSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSGSHQFEQLSGSILW CC ATOM KSIIHRDLKSNNIFLHEDLTVKIGDFGLATVK-----------LSGSILW CC ******************************** ******* CC SEQRES MAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMV CC ATOM MAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMV CC ************************************************** CC SEQRES GRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLAR CC ATOM GRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLAR CC ************************************************** CC SEQRES SLPKIHR CC ATOM SLPK--- CC **** SQ SEQUENCE 307 AA; MW; CN; MDRGSHHHHH HGSEDRNRMK TLGRRDSSDD WEIPDGQITV GQRIGSGSFG TVYKGKWHGD VAVKMLNVTA PTPQQLQAFK NEVGVLRKTR HVNILLFMGY STKPQLAIVT QWCEGSSLYH HLHIIETKFE MIKLIDIARQ TAQGMDYLHA KSIIHRDLKS NNIFLHEDLT VKIGDFGLAT VKSRWSGSHQ FEQLSGSILW MAPEVIRMQD KNPYSFQSDV YAFGIVLYEL MTGQLPYSNI NNRDQIIFMV GRGYLSPDLS KVRSNCPKAM KRLMAECLKK KRDERPLFPQ ILASIELLAR SLPKIHR // ID 4G9CB STANDARD; PRT; 307 AA. DT CONVERTED FROM PDB (SEQRES) 4G9C DE Serine/threonine-protein kinase B-raf OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 3.500 CC R-Factor 0.262 FT #SUB 29 448 ASP B 87 506 ARG A Protein S 8 FT #SUB 29 448 ASP B 88 507 LYS A Protein S 1 FT #SUB 30 449 ASP B 151 570 LYS A Protein B 1 FT #SUB 31 450 TRP B 87 506 ARG A Protein S 2 FT #SUB 31 450 TRP B 88 507 LYS A Protein S 3 FT #SUB 31 450 TRP B 90 509 ARG A Protein S 9 FT #SUB 31 450 TRP B 147 566 TYR A Protein S 1 FT #SUB 56 475 LYS B 296 715 GLU A Protein S 1 FT #SUB 57 476 TRP B 147 566 TYR A Protein S 2 FT #SUB 58 477 HIS B 91 510 HIS A Protein A 6 FT #SUB 58 477 HIS B 143 562 GLN A Protein A 8 FT #SUB 58 477 HIS B 146 565 ASP A Protein S 7 FT #SUB 58 477 HIS B 147 566 TYR A Protein S 4 FT #SUB 58 477 HIS B 150 569 ALA A Protein S 2 FT #SUB 59 478 GLY B 143 562 GLN A Protein B 7 FT #SUB 86 505 LEU B 90 509 ARG A Protein B 1 FT #SUB 87 506 ARG B 29 448 ASP A Protein S 6 FT #SUB 87 506 ARG B 31 450 TRP A Protein B 2 FT #SUB 87 506 ARG B 90 509 ARG A Protein B 1 FT #SUB 88 507 LYS B 29 448 ASP A Protein S 1 FT #SUB 88 507 LYS B 31 450 TRP A Protein B 2 FT #SUB 89 508 THR B 90 509 ARG A Protein B 3 FT #SUB 90 509 ARG B 31 450 TRP A Protein S 7 FT #SUB 90 509 ARG B 86 505 LEU A Protein S 1 FT #SUB 90 509 ARG B 87 506 ARG A Protein S 1 FT #SUB 90 509 ARG B 89 508 THR A Protein S 3 FT #SUB 90 509 ARG B 90 509 ARG A Protein S 8 FT #SUB 90 509 ARG B 96 515 LEU A Protein S 3 FT #SUB 90 509 ARG B 97 516 PHE A Protein S 12 FT #SUB 90 509 ARG B 98 517 MET A Protein B 1 FT #SUB 91 510 HIS B 58 477 HIS A Protein S 2 FT #SUB 91 510 HIS B 96 515 LEU A Protein B 1 FT #SUB 96 515 LEU B 90 509 ARG A Protein S 2 FT #SUB 96 515 LEU B 91 510 HIS A Protein S 2 FT #SUB 97 516 PHE B 90 509 ARG A Protein A 8 FT #SUB 98 517 MET B 90 509 ARG A Protein S 3 FT #SUB 98 517 MET B 91 510 HIS A Protein S 1 FT #SUB 143 562 GLN B 58 477 HIS A Protein S 4 FT #SUB 143 562 GLN B 59 478 GLY A Protein S 5 FT #SUB 146 565 ASP B 58 477 HIS A Protein S 3 FT #SUB 147 566 TYR B 57 476 TRP A Protein S 1 FT #SUB 150 569 ALA B 58 477 HIS A Protein S 2 FT #SUB 167 586 GLU B 169 588 LEU A Protein S 1 FT #SUB 169 588 LEU B 167 586 GLU A Protein S 1 FT #HET 44 463 ILE B 2 801 0WP B S 2 FT #HET 62 481 ALA B 2 801 0WP B A 6 FT #HET 64 483 LYS B 2 801 0WP B A 3 FT #HET 82 501 GLU B 2 801 0WP B S 10 FT #HET 85 504 VAL B 2 801 0WP B S 1 FT #HET 86 505 LEU B 2 801 0WP B S 3 FT #HET 95 514 LEU B 2 801 0WP B S 6 FT #HET 108 527 ILE B 2 801 0WP B A 5 FT #HET 110 529 THR B 2 801 0WP B S 14 FT #HET 111 530 GLN B 2 801 0WP B B 2 FT #HET 112 531 TRP B 2 801 0WP B A 17 FT #HET 113 532 CYS B 2 801 0WP B A 12 FT #HET 154 573 ILE B 2 801 0WP B B 1 FT #HET 155 574 HIS B 2 801 0WP B A 9 FT #HET 164 583 PHE B 2 801 0WP B S 6 FT #HET 174 593 GLY B 2 801 0WP B B 3 FT #HET 175 594 ASP B 2 801 0WP B A 11 FT #HET 176 595 PHE B 2 801 0WP B A 17 FT DISORDER 1 28 FT DISORDER 182 193 FT DISORDER 305 307 CC SEQUENCE 264 AA (ATOM); CC DDWEIPDGQI TVGQRIGSGS FGTVYKGKWH GDVAVKMLNV TAPTPQQLQA FKNEVGVLRK CC TRHVNILLFM GYSTKPQLAI VTQWCEGSSL YHHLHIIETK FEMIKLIDIA RQTAQGMDYL CC HAKSIIHRDL KSNNIFLHED LTVKIGDFGL ATVLSGSILW MAPEVIRMQD KNPYSFQSDV CC YAFGIVLYEL MTGQLPYSNI NNRDQIIFMV GRGYLSPDLS KVRSNCPKAM KRLMAECLKK CC KRDERPLFPQ ILASIELLAR SLPK CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES MDRGSHHHHHHGSEDRNRMKTLGRRDSSDDWEIPDGQITVGQRIGSGSFG CC ATOM ----------------------------DDWEIPDGQITVGQRIGSGSFG CC ********************** CC SEQRES TVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGY CC ATOM TVYKGKWHGDVAVKMLNVTAPTPQQLQAFKNEVGVLRKTRHVNILLFMGY CC ************************************************** CC SEQRES STKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHA CC ATOM STKPQLAIVTQWCEGSSLYHHLHIIETKFEMIKLIDIARQTAQGMDYLHA CC ************************************************** CC SEQRES KSIIHRDLKSNNIFLHEDLTVKIGDFGLATVKSRWSGSHQFEQLSGSILW CC ATOM KSIIHRDLKSNNIFLHEDLTVKIGDFGLATV------------LSGSILW CC ******************************* ******* CC SEQRES MAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMV CC ATOM MAPEVIRMQDKNPYSFQSDVYAFGIVLYELMTGQLPYSNINNRDQIIFMV CC ************************************************** CC SEQRES GRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLAR CC ATOM GRGYLSPDLSKVRSNCPKAMKRLMAECLKKKRDERPLFPQILASIELLAR CC ************************************************** CC SEQRES SLPKIHR CC ATOM SLPK--- CC **** SQ SEQUENCE 307 AA; MW; CN; MDRGSHHHHH HGSEDRNRMK TLGRRDSSDD WEIPDGQITV GQRIGSGSFG TVYKGKWHGD VAVKMLNVTA PTPQQLQAFK NEVGVLRKTR HVNILLFMGY STKPQLAIVT QWCEGSSLYH HLHIIETKFE MIKLIDIARQ TAQGMDYLHA KSIIHRDLKS NNIFLHEDLT VKIGDFGLAT VKSRWSGSHQ FEQLSGSILW MAPEVIRMQD KNPYSFQSDV YAFGIVLYEL MTGQLPYSNI NNRDQIIFMV GRGYLSPDLS KVRSNCPKAM KRLMAECLKK KRDERPLFPQ ILASIELLAR SLPKIHR //