ID 3RQDA STANDARD; PRT; 389 AA. DT CONVERTED FROM PDB (SEQRES) 3RQD DE Histone deacetylase 8 OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.140 CC R-Factor 0.204 FT #SUB 32 32 ALA A 100 100 TYR B Protein B 3 FT #SUB 33 33 LYS A 100 100 TYR B Protein B 1 FT #SUB 35 35 PRO A 100 100 TYR B Protein S 2 FT #SUB 100 100 TYR A 32 32 ALA B Protein B 3 FT #SUB 100 100 TYR A 33 33 LYS B Protein B 1 FT #SUB 100 100 TYR A 35 35 PRO B Protein S 2 FT #SUB 100 100 TYR A 308 308 LEU B Protein S 1 FT #SUB 205 205 PRO A 275 275 CYS B Protein B 1 FT #SUB 205 205 PRO A 353 353 ARG B Protein B 2 FT #SUB 206 206 GLY A 275 275 CYS B Protein B 5 FT #SUB 275 275 CYS A 205 205 PRO B Protein S 1 FT #SUB 275 275 CYS A 206 206 GLY B Protein S 5 FT #SUB 275 275 CYS A 207 207 PHE B Protein S 1 FT #SUB 308 308 LEU A 100 100 TYR B Protein S 1 FT #SUB 353 353 ARG A 205 205 PRO B Protein S 2 FT #SUB 356 356 ARG A 356 356 ARG B Protein S 1 FT #SUB 101 101 ASP A 1 1 02G C Protein S 2 FT #SUB 101 101 ASP A 2 2 GLY C Protein S 6 FT #SUB 101 101 ASP A 3 3 BB9 C Protein S 3 FT #SUB 101 101 ASP A 4 4 03Y C Protein A 3 FT #SUB 142 142 HIS A 1 1 02G C Protein S 1 FT #SUB 143 143 HIS A 1 1 02G C Protein S 3 FT #SUB 151 151 GLY A 1 1 02G C Protein B 2 FT #SUB 152 152 PHE A 1 1 02G C Protein S 6 FT #SUB 178 178 ASP A 1 1 02G C Protein S 2 FT #SUB 180 180 HIS A 1 1 02G C Protein S 8 FT #SUB 208 208 PHE A 1 1 02G C Protein S 13 FT #SUB 208 208 PHE A 2 2 GLY C Protein S 3 FT #SUB 267 267 ASP A 1 1 02G C Protein S 1 FT #SUB 274 274 MET A 1 1 02G C Protein S 2 FT #SUB 274 274 MET A 5 5 VAL C Protein S 2 FT #SUB 304 304 GLY A 1 1 02G C Protein B 1 FT #SUB 306 306 TYR A 1 1 02G C Protein S 3 FT #SUB 152 152 PHE A 4 4 03Y D Protein S 3 FT #SUB 273 273 PRO A 3 3 BB9 D Protein S 1 FT #SUB 273 273 PRO A 5 5 VAL D Protein A 3 FT #SUB 274 274 MET A 5 5 VAL D Protein S 2 FT #SUB 306 306 TYR A 4 4 03Y D Protein S 1 FT #HET 176 176 ASP A 2 402 K A A 5 FT #HET 178 178 ASP A 1 401 ZN A S 3 FT #HET 178 178 ASP A 2 402 K A B 3 FT #HET 180 180 HIS A 1 401 ZN A A 5 FT #HET 180 180 HIS A 2 402 K A B 2 FT #HET 189 189 PHE A 3 403 K A B 2 FT #HET 192 192 THR A 3 403 K A B 1 FT #HET 195 195 VAL A 3 403 K A B 1 FT #HET 199 199 SER A 2 402 K A S 1 FT #HET 200 200 LEU A 2 402 K A B 2 FT #HET 201 201 HIS A 2 402 K A S 1 FT #HET 225 225 TYR A 3 403 K A A 3 FT #HET 267 267 ASP A 1 401 ZN A S 3 FT DISORDER 1 13 FT DISORDER 85 94 FT DISORDER 378 389 CC SEQUENCE 354 AA (ATOM); CC LVPVYIYSPE YVSMCDSLAK IPKRASMVHS LIEAYALHKQ MRIVKPKVAS MEEMATFHTD CC AYLQHLQKVS QEYGLGYDCP ATEGIFDYAA AIGGATITAA QCLIDGMCKV AINWSGGWHH CC AKKDEASGFC YLNDAVLGIL RLRRKFERIL YVDLDLHHGD GVEDAFSFTS KVMTVSLHKF CC SPGFFPGTGD VSDVGLGKGR YYSVNVPIQD GIQDEKYYQI CESVLKEVYQ AFNPKAVVLQ CC LGADTIAGDP MCSFNMTPVG IGKCLKYILQ WQLATLILGG GGYNLANTAR CWTYLTGVIL CC GKTLSSEIPD HEFFTAYGPD YVLEITPSCR PDRNEPHRIQ QILNYIKGNL KHVV CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES MEEPEEPADSGQSLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYAL CC ATOM -------------LVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYAL CC ************************************* CC SEQRES HKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGY CC ATOM HKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQ----------EYGLGY CC ********************************** ****** CC SEQRES DCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEAS CC ATOM DCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEAS CC ************************************************** CC SEQRES GFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSL CC ATOM GFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSL CC ************************************************** CC SEQRES HKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKE CC ATOM HKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKE CC ************************************************** CC SEQRES VYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLI CC ATOM VYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLI CC ************************************************** CC SEQRES LGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITP CC ATOM LGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITP CC ************************************************** CC SEQRES SCRPDRNEPHRIQQILNYIKGNLKHVVIEGRGSHHHHHH CC ATOM SCRPDRNEPHRIQQILNYIKGNLKHVV------------ CC *************************** SQ SEQUENCE 389 AA; MW; CN; MEEPEEPADS GQSLVPVYIY SPEYVSMCDS LAKIPKRASM VHSLIEAYAL HKQMRIVKPK VASMEEMATF HTDAYLQHLQ KVSQEGDDDH PDSIEYGLGY DCPATEGIFD YAAAIGGATI TAAQCLIDGM CKVAINWSGG WHHAKKDEAS GFCYLNDAVL GILRLRRKFE RILYVDLDLH HGDGVEDAFS FTSKVMTVSL HKFSPGFFPG TGDVSDVGLG KGRYYSVNVP IQDGIQDEKY YQICESVLKE VYQAFNPKAV VLQLGADTIA GDPMCSFNMT PVGIGKCLKY ILQWQLATLI LGGGGYNLAN TARCWTYLTG VILGKTLSSE IPDHEFFTAY GPDYVLEITP SCRPDRNEPH RIQQILNYIK GNLKHVVIEG RGSHHHHHH // ID 3RQDB STANDARD; PRT; 389 AA. DT CONVERTED FROM PDB (SEQRES) 3RQD DE Histone deacetylase 8 OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.140 CC R-Factor 0.204 FT #SUB 32 32 ALA B 100 100 TYR A Protein B 3 FT #SUB 33 33 LYS B 100 100 TYR A Protein B 1 FT #SUB 35 35 PRO B 100 100 TYR A Protein S 2 FT #SUB 100 100 TYR B 32 32 ALA A Protein B 3 FT #SUB 100 100 TYR B 33 33 LYS A Protein B 1 FT #SUB 100 100 TYR B 35 35 PRO A Protein S 2 FT #SUB 100 100 TYR B 308 308 LEU A Protein S 1 FT #SUB 205 205 PRO B 275 275 CYS A Protein B 1 FT #SUB 205 205 PRO B 353 353 ARG A Protein B 2 FT #SUB 206 206 GLY B 275 275 CYS A Protein B 5 FT #SUB 207 207 PHE B 275 275 CYS A Protein B 1 FT #SUB 275 275 CYS B 205 205 PRO A Protein S 1 FT #SUB 275 275 CYS B 206 206 GLY A Protein S 5 FT #SUB 308 308 LEU B 100 100 TYR A Protein S 1 FT #SUB 353 353 ARG B 205 205 PRO A Protein S 2 FT #SUB 356 356 ARG B 356 356 ARG A Protein S 1 FT #SUB 152 152 PHE B 4 4 03Y C Protein S 3 FT #SUB 273 273 PRO B 3 3 BB9 C Protein S 1 FT #SUB 273 273 PRO B 5 5 VAL C Protein A 2 FT #SUB 274 274 MET B 5 5 VAL C Protein S 2 FT #SUB 100 100 TYR B 4 4 03Y D Protein B 1 FT #SUB 101 101 ASP B 1 1 02G D Protein S 2 FT #SUB 101 101 ASP B 2 2 GLY D Protein S 6 FT #SUB 101 101 ASP B 3 3 BB9 D Protein S 2 FT #SUB 101 101 ASP B 4 4 03Y D Protein A 3 FT #SUB 142 142 HIS B 1 1 02G D Protein S 1 FT #SUB 143 143 HIS B 1 1 02G D Protein S 3 FT #SUB 151 151 GLY B 1 1 02G D Protein B 2 FT #SUB 152 152 PHE B 1 1 02G D Protein S 3 FT #SUB 178 178 ASP B 1 1 02G D Protein S 2 FT #SUB 180 180 HIS B 1 1 02G D Protein S 9 FT #SUB 208 208 PHE B 1 1 02G D Protein S 13 FT #SUB 208 208 PHE B 2 2 GLY D Protein S 3 FT #SUB 267 267 ASP B 1 1 02G D Protein S 1 FT #SUB 274 274 MET B 1 1 02G D Protein S 2 FT #SUB 274 274 MET B 5 5 VAL D Protein S 2 FT #SUB 304 304 GLY B 1 1 02G D Protein B 1 FT #SUB 306 306 TYR B 1 1 02G D Protein S 3 FT #HET 176 176 ASP B 5 402 K B A 5 FT #HET 177 177 LEU B 5 402 K B B 1 FT #HET 178 178 ASP B 4 401 ZN B S 3 FT #HET 178 178 ASP B 5 402 K B B 4 FT #HET 180 180 HIS B 4 401 ZN B A 5 FT #HET 180 180 HIS B 5 402 K B B 2 FT #HET 189 189 PHE B 6 403 K B B 2 FT #HET 192 192 THR B 6 403 K B B 1 FT #HET 195 195 VAL B 6 403 K B B 2 FT #HET 199 199 SER B 5 402 K B S 1 FT #HET 200 200 LEU B 5 402 K B B 3 FT #HET 201 201 HIS B 5 402 K B S 1 FT #HET 225 225 TYR B 6 403 K B A 3 FT #HET 267 267 ASP B 4 401 ZN B S 3 FT DISORDER 1 12 FT DISORDER 84 93 FT DISORDER 379 389 CC SEQUENCE 356 AA (ATOM); CC SLVPVYIYSP EYVSMCDSLA KIPKRASMVH SLIEAYALHK QMRIVKPKVA SMEEMATFHT CC DAYLQHLQKV SIEYGLGYDC PATEGIFDYA AAIGGATITA AQCLIDGMCK VAINWSGGWH CC HAKKDEASGF CYLNDAVLGI LRLRRKFERI LYVDLDLHHG DGVEDAFSFT SKVMTVSLHK CC FSPGFFPGTG DVSDVGLGKG RYYSVNVPIQ DGIQDEKYYQ ICESVLKEVY QAFNPKAVVL CC QLGADTIAGD PMCSFNMTPV GIGKCLKYIL QWQLATLILG GGGYNLANTA RCWTYLTGVI CC LGKTLSSEIP DHEFFTAYGP DYVLEITPSC RPDRNEPHRI QQILNYIKGN LKHVVI CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES MEEPEEPADSGQSLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYAL CC ATOM ------------SLVPVYIYSPEYVSMCDSLAKIPKRASMVHSLIEAYAL CC ************************************** CC SEQRES HKQMRIVKPKVASMEEMATFHTDAYLQHLQKVSQEGDDDHPDSIEYGLGY CC ATOM HKQMRIVKPKVASMEEMATFHTDAYLQHLQKVS----------IEYGLGY CC ********************************* ******* CC SEQRES DCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEAS CC ATOM DCPATEGIFDYAAAIGGATITAAQCLIDGMCKVAINWSGGWHHAKKDEAS CC ************************************************** CC SEQRES GFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSL CC ATOM GFCYLNDAVLGILRLRRKFERILYVDLDLHHGDGVEDAFSFTSKVMTVSL CC ************************************************** CC SEQRES HKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKE CC ATOM HKFSPGFFPGTGDVSDVGLGKGRYYSVNVPIQDGIQDEKYYQICESVLKE CC ************************************************** CC SEQRES VYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLI CC ATOM VYQAFNPKAVVLQLGADTIAGDPMCSFNMTPVGIGKCLKYILQWQLATLI CC ************************************************** CC SEQRES LGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITP CC ATOM LGGGGYNLANTARCWTYLTGVILGKTLSSEIPDHEFFTAYGPDYVLEITP CC ************************************************** CC SEQRES SCRPDRNEPHRIQQILNYIKGNLKHVVIEGRGSHHHHHH CC ATOM SCRPDRNEPHRIQQILNYIKGNLKHVVI----------- CC **************************** SQ SEQUENCE 389 AA; MW; CN; MEEPEEPADS GQSLVPVYIY SPEYVSMCDS LAKIPKRASM VHSLIEAYAL HKQMRIVKPK VASMEEMATF HTDAYLQHLQ KVSQEGDDDH PDSIEYGLGY DCPATEGIFD YAAAIGGATI TAAQCLIDGM CKVAINWSGG WHHAKKDEAS GFCYLNDAVL GILRLRRKFE RILYVDLDLH HGDGVEDAFS FTSKVMTVSL HKFSPGFFPG TGDVSDVGLG KGRYYSVNVP IQDGIQDEKY YQICESVLKE VYQAFNPKAV VLQLGADTIA GDPMCSFNMT PVGIGKCLKY ILQWQLATLI LGGGGYNLAN TARCWTYLTG VILGKTLSSE IPDHEFFTAY GPDYVLEITP SCRPDRNEPH RIQQILNYIK GNLKHVVIEG RGSHHHHHH // ID 3RQDC STANDARD; PRT; 5 AA. DT CONVERTED FROM PDB (SEQRES) 3RQD DE Largazole OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.140 CC R-Factor 0.204 FT #SUB 1 1 02G C 101 101 ASP A Protein A 2 FT #SUB 1 1 02G C 142 142 HIS A Protein S 1 FT #SUB 1 1 02G C 143 143 HIS A Protein S 3 FT #SUB 1 1 02G C 151 151 GLY A Protein S 2 FT #SUB 1 1 02G C 152 152 PHE A Protein S 6 FT #SUB 1 1 02G C 178 178 ASP A Protein S 2 FT #SUB 1 1 02G C 180 180 HIS A Protein S 8 FT #SUB 1 1 02G C 208 208 PHE A Protein A 13 FT #SUB 1 1 02G C 267 267 ASP A Protein S 1 FT #SUB 1 1 02G C 274 274 MET A Protein S 2 FT #SUB 1 1 02G C 304 304 GLY A Protein S 1 FT #SUB 1 1 02G C 306 306 TYR A Protein S 3 FT #SUB 2 2 GLY C 101 101 ASP A Protein B 6 FT #SUB 2 2 GLY C 208 208 PHE A Protein B 3 FT #SUB 3 3 BB9 C 101 101 ASP A Protein B 3 FT #SUB 4 4 03Y C 101 101 ASP A Protein B 3 FT #SUB 5 5 VAL C 274 274 MET A Protein B 2 FT #SUB 3 3 BB9 C 273 273 PRO B Protein S 1 FT #SUB 4 4 03Y C 152 152 PHE B Protein A 3 FT #SUB 5 5 VAL C 273 273 PRO B Protein S 2 FT #SUB 5 5 VAL C 274 274 MET B Protein S 2 FT #SUB 4 4 03Y C 4 4 03Y D Protein A 4 FT #SUB 4 4 03Y C 5 5 VAL D Protein B 3 FT #SUB 5 5 VAL C 4 4 03Y D Protein B 3 FT #SUB 5 5 VAL C 5 5 VAL D Protein A 2 FT #HET 1 1 02G C 1 401 ZN A S 3 CC Miss-BB 1 CC SEQUENCE 5 AA (ATOM); CC XGXXV CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XGXXV CC ATOM XGXXV CC ***** SQ SEQUENCE 5 AA; MW; CN; XGXXV // ID 3RQDD STANDARD; PRT; 5 AA. DT CONVERTED FROM PDB (SEQRES) 3RQD DE Largazole OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 2.140 CC R-Factor 0.204 FT #SUB 3 3 BB9 D 273 273 PRO A Protein S 1 FT #SUB 4 4 03Y D 152 152 PHE A Protein A 3 FT #SUB 4 4 03Y D 306 306 TYR A Protein S 1 FT #SUB 5 5 VAL D 273 273 PRO A Protein S 3 FT #SUB 5 5 VAL D 274 274 MET A Protein S 2 FT #SUB 1 1 02G D 101 101 ASP B Protein A 2 FT #SUB 1 1 02G D 142 142 HIS B Protein S 1 FT #SUB 1 1 02G D 143 143 HIS B Protein S 3 FT #SUB 1 1 02G D 151 151 GLY B Protein S 2 FT #SUB 1 1 02G D 152 152 PHE B Protein S 3 FT #SUB 1 1 02G D 178 178 ASP B Protein S 2 FT #SUB 1 1 02G D 180 180 HIS B Protein S 9 FT #SUB 1 1 02G D 208 208 PHE B Protein A 13 FT #SUB 1 1 02G D 267 267 ASP B Protein S 1 FT #SUB 1 1 02G D 274 274 MET B Protein S 2 FT #SUB 1 1 02G D 304 304 GLY B Protein S 1 FT #SUB 1 1 02G D 306 306 TYR B Protein S 3 FT #SUB 2 2 GLY D 101 101 ASP B Protein B 6 FT #SUB 2 2 GLY D 208 208 PHE B Protein B 3 FT #SUB 3 3 BB9 D 101 101 ASP B Protein B 2 FT #SUB 4 4 03Y D 100 100 TYR B Protein S 1 FT #SUB 4 4 03Y D 101 101 ASP B Protein B 3 FT #SUB 5 5 VAL D 274 274 MET B Protein B 2 FT #SUB 4 4 03Y D 4 4 03Y C Protein A 4 FT #SUB 4 4 03Y D 5 5 VAL C Protein B 3 FT #SUB 5 5 VAL D 4 4 03Y C Protein B 3 FT #SUB 5 5 VAL D 5 5 VAL C Protein A 2 FT #HET 1 1 02G D 4 401 ZN B S 3 CC Miss-BB 1 CC SEQUENCE 5 AA (ATOM); CC XGXXV CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES XGXXV CC ATOM XGXXV CC ***** SQ SEQUENCE 5 AA; MW; CN; XGXXV //