ID 1XQHA STANDARD; PRT; 264 AA. DT CONVERTED FROM PDB (SEQRES) 1XQH DE Histone-lysine N-methyltransferase, H3 lysine-4 specific OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 1.750 CC R-Factor 0.186 FT #SUB 143 245 TYR A 4 372 MLZ B Protein S 6 FT #SUB 153 255 VAL A 2 370 LYS B Protein S 2 FT #SUB 154 256 ASP A 1 369 LEU B Protein S 5 FT #SUB 154 256 ASP A 2 370 LYS B Protein A 3 FT #SUB 156 258 ARG A 2 370 LYS B Protein B 4 FT #SUB 158 260 TRP A 2 370 LYS B Protein S 11 FT #SUB 161 263 ASN A 2 370 LYS B Protein S 5 FT #SUB 162 264 GLY A 4 372 MLZ B Protein B 2 FT #SUB 163 265 ASN A 4 372 MLZ B Protein S 1 FT #SUB 164 266 THR A 2 370 LYS B Protein S 3 FT #SUB 164 266 THR A 3 371 SER B Protein A 7 FT #SUB 164 266 THR A 4 372 MLZ B Protein B 6 FT #SUB 165 267 LEU A 4 372 MLZ B Protein A 6 FT #SUB 166 268 SER A 3 371 SER B Protein A 4 FT #SUB 166 268 SER A 4 372 MLZ B Protein A 5 FT #SUB 191 293 HIS A 4 372 MLZ B Protein B 1 FT #SUB 203 305 TYR A 4 372 MLZ B Protein S 6 FT #SUB 215 317 LYS A 6 374 GLY B Protein S 1 FT #SUB 233 335 TYR A 4 372 MLZ B Protein A 12 FT #SUB 233 335 TYR A 5 373 LYS B Protein B 3 FT #SUB 234 336 GLY A 5 373 LYS B Protein B 2 FT #SUB 235 337 TYR A 3 371 SER B Protein S 3 FT #SUB 235 337 TYR A 4 372 MLZ B Protein S 3 FT #SUB 246 348 GLU A 2 370 LYS B Protein S 2 FT #SUB 15 117 GLY A 20 122 TYR E Protein B 2 FT #SUB 16 118 VAL A 18 120 TRP E Protein B 1 FT #SUB 16 118 VAL A 19 121 ILE E Protein B 2 FT #SUB 16 118 VAL A 20 122 TYR E Protein B 5 FT #SUB 17 119 CYS A 17 119 CYS E Protein S 1 FT #SUB 17 119 CYS A 18 120 TRP E Protein A 4 FT #SUB 17 119 CYS A 19 121 ILE E Protein S 1 FT #SUB 18 120 TRP A 16 118 VAL E Protein B 1 FT #SUB 18 120 TRP A 17 119 CYS E Protein B 4 FT #SUB 18 120 TRP A 18 120 TRP E Protein B 7 FT #SUB 18 120 TRP A 20 122 TYR E Protein S 4 FT #SUB 19 121 ILE A 16 118 VAL E Protein B 2 FT #SUB 19 121 ILE A 17 119 CYS E Protein S 1 FT #SUB 20 122 TYR A 15 117 GLY E Protein B 2 FT #SUB 20 122 TYR A 16 118 VAL E Protein A 5 FT #SUB 20 122 TYR A 18 120 TRP E Protein S 2 FT #SUB 20 122 TYR A 75 177 GLU E Protein S 4 FT #SUB 20 122 TYR A 76 178 GLY E Protein S 8 FT #SUB 22 124 PRO A 77 179 ARG E Protein B 1 FT #SUB 24 126 GLY A 75 177 GLU E Protein B 3 FT #SUB 49 151 GLU A 75 177 GLU E Protein S 1 FT #SUB 75 177 GLU A 20 122 TYR E Protein B 5 FT #SUB 75 177 GLU A 24 126 GLY E Protein S 4 FT #SUB 75 177 GLU A 49 151 GLU E Protein B 1 FT #SUB 76 178 GLY A 20 122 TYR E Protein B 8 FT #SUB 77 179 ARG A 22 124 PRO E Protein S 1 FT #HET 121 223 ILE A 1 1501 SAH A S 1 FT #HET 124 226 ALA A 1 1501 SAH A A 7 FT #HET 125 227 GLY A 1 1501 SAH A B 1 FT #HET 126 228 GLU A 1 1501 SAH A A 19 FT #HET 162 264 GLY A 1 1501 SAH A B 1 FT #HET 163 265 ASN A 1 1501 SAH A S 2 FT #HET 191 293 HIS A 1 1501 SAH A B 3 FT #HET 192 294 LYS A 1 1501 SAH A A 9 FT #HET 193 295 ALA A 1 1501 SAH A B 1 FT #HET 194 296 ASN A 1 1501 SAH A A 16 FT #HET 195 297 HIS A 1 1501 SAH A A 6 FT #HET 233 335 TYR A 1 1501 SAH A S 7 FT #HET 250 352 TRP A 1 1501 SAH A S 23 FT #HET 254 356 GLU A 1 1501 SAH A S 5 FT DISORDER 1 14 CC SEQUENCE 250 AA (ATOM); CC GVCWIYYPDG GSLVGEVNED GEMTGEKIAY VYPDERTALY GKFIDGEMIE GKLATLMSTE CC EGRPHFELMP GNSVYHFDKS TSSCISTNAL LPDPYESERV YVAESLISSA GEGLFSKVAV CC GPNTVMSFYN GVRITHQEVD SRDWALNGNT LSLDEETVID VPEPYNHVSK YCASLGHKAN CC HSFTPNCIYD MFVHPRFGPI KCIRTLRAVE ADEELTVAYG YDHSPPGKSG PEAPEWYQVE CC LKAFQATQQK CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES GPLGSGQYKDNIRHGVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDER CC ATOM --------------GVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDER CC ************************************ CC SEQRES TALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCIS CC ATOM TALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCIS CC ************************************************** CC SEQRES TNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITH CC ATOM TNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITH CC ************************************************** CC SEQRES QEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPN CC ATOM QEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPN CC ************************************************** CC SEQRES CIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGYDHSPPGKSGPEAPEW CC ATOM CIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGYDHSPPGKSGPEAPEW CC ************************************************** CC SEQRES YQVELKAFQATQQK CC ATOM YQVELKAFQATQQK CC ************** SQ SEQUENCE 264 AA; MW; CN; GPLGSGQYKD NIRHGVCWIY YPDGGSLVGE VNEDGEMTGE KIAYVYPDER TALYGKFIDG EMIEGKLATL MSTEEGRPHF ELMPGNSVYH FDKSTSSCIS TNALLPDPYE SERVYVAESL ISSAGEGLFS KVAVGPNTVM SFYNGVRITH QEVDSRDWAL NGNTLSLDEE TVIDVPEPYN HVSKYCASLG HKANHSFTPN CIYDMFVHPR FGPIKCIRTL RAVEADEELT VAYGYDHSPP GKSGPEAPEW YQVELKAFQA TQQK // ID 1XQHB STANDARD; PRT; 10 AA. DT CONVERTED FROM PDB (SEQRES) 1XQH DE 9-mer peptide from tumor protein p53 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 1.750 CC R-Factor 0.186 FT #SUB 1 369 LEU B 154 256 ASP A Protein A 5 FT #SUB 2 370 LYS B 153 255 VAL A Protein B 2 FT #SUB 2 370 LYS B 154 256 ASP A Protein A 3 FT #SUB 2 370 LYS B 156 258 ARG A Protein S 4 FT #SUB 2 370 LYS B 158 260 TRP A Protein A 11 FT #SUB 2 370 LYS B 161 263 ASN A Protein A 5 FT #SUB 2 370 LYS B 164 266 THR A Protein B 3 FT #SUB 2 370 LYS B 246 348 GLU A Protein S 2 FT #SUB 3 371 SER B 164 266 THR A Protein A 7 FT #SUB 3 371 SER B 166 268 SER A Protein S 4 FT #SUB 3 371 SER B 235 337 TYR A Protein B 3 FT #SUB 4 372 MLZ B 143 245 TYR A Protein S 6 FT #SUB 4 372 MLZ B 162 264 GLY A Protein S 2 FT #SUB 4 372 MLZ B 163 265 ASN A Protein S 1 FT #SUB 4 372 MLZ B 164 266 THR A Protein A 6 FT #SUB 4 372 MLZ B 165 267 LEU A Protein A 6 FT #SUB 4 372 MLZ B 166 268 SER A Protein B 5 FT #SUB 4 372 MLZ B 191 293 HIS A Protein S 1 FT #SUB 4 372 MLZ B 203 305 TYR A Protein S 6 FT #SUB 4 372 MLZ B 233 335 TYR A Protein A 12 FT #SUB 4 372 MLZ B 235 337 TYR A Protein A 3 FT #SUB 5 373 LYS B 233 335 TYR A Protein B 3 FT #SUB 5 373 LYS B 234 336 GLY A Protein A 2 FT #SUB 6 374 GLY B 215 317 LYS A Protein B 1 FT #HET 4 372 MLZ B 1 1501 SAH A S 2 FT DISORDER 7 10 CC SEQUENCE 6 AA (ATOM); CC LKSXKG CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES LKSXKGQSTY CC ATOM LKSXKG---- CC ****** SQ SEQUENCE 10 AA; MW; CN; LKSXKGQSTY // ID 1XQHE STANDARD; PRT; 264 AA. DT CONVERTED FROM PDB (SEQRES) 1XQH DE Histone-lysine N-methyltransferase, H3 lysine-4 specific OS Homo sapiens CC EXPDTA X-RAY DIFFRACTION CC RESOLU 1.750 CC R-Factor 0.186 FT #SUB 15 117 GLY E 20 122 TYR A Protein B 2 FT #SUB 16 118 VAL E 18 120 TRP A Protein B 1 FT #SUB 16 118 VAL E 19 121 ILE A Protein B 2 FT #SUB 16 118 VAL E 20 122 TYR A Protein B 5 FT #SUB 17 119 CYS E 17 119 CYS A Protein S 1 FT #SUB 17 119 CYS E 18 120 TRP A Protein A 4 FT #SUB 17 119 CYS E 19 121 ILE A Protein S 1 FT #SUB 18 120 TRP E 16 118 VAL A Protein B 1 FT #SUB 18 120 TRP E 17 119 CYS A Protein B 4 FT #SUB 18 120 TRP E 18 120 TRP A Protein B 7 FT #SUB 18 120 TRP E 20 122 TYR A Protein S 2 FT #SUB 19 121 ILE E 16 118 VAL A Protein B 2 FT #SUB 19 121 ILE E 17 119 CYS A Protein S 1 FT #SUB 20 122 TYR E 15 117 GLY A Protein B 2 FT #SUB 20 122 TYR E 16 118 VAL A Protein A 5 FT #SUB 20 122 TYR E 18 120 TRP A Protein S 4 FT #SUB 20 122 TYR E 75 177 GLU A Protein S 5 FT #SUB 20 122 TYR E 76 178 GLY A Protein S 8 FT #SUB 22 124 PRO E 77 179 ARG A Protein B 1 FT #SUB 24 126 GLY E 75 177 GLU A Protein B 4 FT #SUB 49 151 GLU E 75 177 GLU A Protein S 1 FT #SUB 75 177 GLU E 20 122 TYR A Protein B 4 FT #SUB 75 177 GLU E 24 126 GLY A Protein S 3 FT #SUB 75 177 GLU E 49 151 GLU A Protein B 1 FT #SUB 76 178 GLY E 20 122 TYR A Protein B 8 FT #SUB 77 179 ARG E 22 124 PRO A Protein S 1 FT #SUB 143 245 TYR E 4 372 MLZ F Protein S 5 FT #SUB 153 255 VAL E 2 370 LYS F Protein A 4 FT #SUB 154 256 ASP E 1 369 LEU F Protein S 5 FT #SUB 154 256 ASP E 2 370 LYS F Protein A 3 FT #SUB 156 258 ARG E 2 370 LYS F Protein B 4 FT #SUB 158 260 TRP E 1 369 LEU F Protein S 1 FT #SUB 158 260 TRP E 2 370 LYS F Protein S 11 FT #SUB 161 263 ASN E 2 370 LYS F Protein S 6 FT #SUB 162 264 GLY E 4 372 MLZ F Protein B 2 FT #SUB 163 265 ASN E 4 372 MLZ F Protein S 1 FT #SUB 164 266 THR E 2 370 LYS F Protein S 3 FT #SUB 164 266 THR E 3 371 SER F Protein A 7 FT #SUB 164 266 THR E 4 372 MLZ F Protein B 6 FT #SUB 165 267 LEU E 4 372 MLZ F Protein A 6 FT #SUB 166 268 SER E 3 371 SER F Protein A 5 FT #SUB 166 268 SER E 4 372 MLZ F Protein A 5 FT #SUB 191 293 HIS E 4 372 MLZ F Protein B 1 FT #SUB 203 305 TYR E 4 372 MLZ F Protein S 5 FT #SUB 215 317 LYS E 6 374 GLY F Protein S 1 FT #SUB 233 335 TYR E 4 372 MLZ F Protein A 14 FT #SUB 233 335 TYR E 5 373 LYS F Protein B 3 FT #SUB 234 336 GLY E 5 373 LYS F Protein B 1 FT #SUB 235 337 TYR E 3 371 SER F Protein S 3 FT #SUB 235 337 TYR E 4 372 MLZ F Protein S 3 FT #SUB 246 348 GLU E 1 369 LEU F Protein B 1 FT #SUB 246 348 GLU E 2 370 LYS F Protein S 1 FT #HET 121 223 ILE E 2 2501 SAH E S 1 FT #HET 124 226 ALA E 2 2501 SAH E A 7 FT #HET 125 227 GLY E 2 2501 SAH E B 2 FT #HET 126 228 GLU E 2 2501 SAH E A 19 FT #HET 162 264 GLY E 2 2501 SAH E B 1 FT #HET 163 265 ASN E 2 2501 SAH E S 2 FT #HET 191 293 HIS E 2 2501 SAH E B 3 FT #HET 192 294 LYS E 2 2501 SAH E A 9 FT #HET 193 295 ALA E 2 2501 SAH E B 1 FT #HET 194 296 ASN E 2 2501 SAH E A 16 FT #HET 195 297 HIS E 2 2501 SAH E A 6 FT #HET 233 335 TYR E 2 2501 SAH E S 5 FT #HET 250 352 TRP E 2 2501 SAH E S 20 FT #HET 254 356 GLU E 2 2501 SAH E S 6 FT DISORDER 1 14 CC SEQUENCE 250 AA (ATOM); CC GVCWIYYPDG GSLVGEVNED GEMTGEKIAY VYPDERTALY GKFIDGEMIE GKLATLMSTE CC EGRPHFELMP GNSVYHFDKS TSSCISTNAL LPDPYESERV YVAESLISSA GEGLFSKVAV CC GPNTVMSFYN GVRITHQEVD SRDWALNGNT LSLDEETVID VPEPYNHVSK YCASLGHKAN CC HSFTPNCIYD MFVHPRFGPI KCIRTLRAVE ADEELTVAYG YDHSPPGKSG PEAPEWYQVE CC LKAFQATQQK CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES GPLGSGQYKDNIRHGVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDER CC ATOM --------------GVCWIYYPDGGSLVGEVNEDGEMTGEKIAYVYPDER CC ************************************ CC SEQRES TALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCIS CC ATOM TALYGKFIDGEMIEGKLATLMSTEEGRPHFELMPGNSVYHFDKSTSSCIS CC ************************************************** CC SEQRES TNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITH CC ATOM TNALLPDPYESERVYVAESLISSAGEGLFSKVAVGPNTVMSFYNGVRITH CC ************************************************** CC SEQRES QEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPN CC ATOM QEVDSRDWALNGNTLSLDEETVIDVPEPYNHVSKYCASLGHKANHSFTPN CC ************************************************** CC SEQRES CIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGYDHSPPGKSGPEAPEW CC ATOM CIYDMFVHPRFGPIKCIRTLRAVEADEELTVAYGYDHSPPGKSGPEAPEW CC ************************************************** CC SEQRES YQVELKAFQATQQK CC ATOM YQVELKAFQATQQK CC ************** SQ SEQUENCE 264 AA; MW; CN; GPLGSGQYKD NIRHGVCWIY YPDGGSLVGE VNEDGEMTGE KIAYVYPDER TALYGKFIDG EMIEGKLATL MSTEEGRPHF ELMPGNSVYH FDKSTSSCIS TNALLPDPYE SERVYVAESL ISSAGEGLFS KVAVGPNTVM SFYNGVRITH QEVDSRDWAL NGNTLSLDEE TVIDVPEPYN HVSKYCASLG HKANHSFTPN CIYDMFVHPR FGPIKCIRTL RAVEADEELT VAYGYDHSPP GKSGPEAPEW YQVELKAFQA TQQK // ID 1XQHF STANDARD; PRT; 10 AA. DT CONVERTED FROM PDB (SEQRES) 1XQH DE 9-mer peptide from tumor protein p53 OS syntetic CC EXPDTA X-RAY DIFFRACTION CC RESOLU 1.750 CC R-Factor 0.186 FT #SUB 1 369 LEU F 154 256 ASP E Protein B 5 FT #SUB 1 369 LEU F 158 260 TRP E Protein B 1 FT #SUB 1 369 LEU F 246 348 GLU E Protein B 1 FT #SUB 2 370 LYS F 153 255 VAL E Protein A 4 FT #SUB 2 370 LYS F 154 256 ASP E Protein A 3 FT #SUB 2 370 LYS F 156 258 ARG E Protein S 4 FT #SUB 2 370 LYS F 158 260 TRP E Protein A 11 FT #SUB 2 370 LYS F 161 263 ASN E Protein A 6 FT #SUB 2 370 LYS F 164 266 THR E Protein B 3 FT #SUB 2 370 LYS F 246 348 GLU E Protein S 1 FT #SUB 3 371 SER F 164 266 THR E Protein A 7 FT #SUB 3 371 SER F 166 268 SER E Protein S 5 FT #SUB 3 371 SER F 235 337 TYR E Protein B 3 FT #SUB 4 372 MLZ F 143 245 TYR E Protein S 5 FT #SUB 4 372 MLZ F 162 264 GLY E Protein S 2 FT #SUB 4 372 MLZ F 163 265 ASN E Protein S 1 FT #SUB 4 372 MLZ F 164 266 THR E Protein A 6 FT #SUB 4 372 MLZ F 165 267 LEU E Protein A 6 FT #SUB 4 372 MLZ F 166 268 SER E Protein B 5 FT #SUB 4 372 MLZ F 191 293 HIS E Protein S 1 FT #SUB 4 372 MLZ F 203 305 TYR E Protein S 5 FT #SUB 4 372 MLZ F 233 335 TYR E Protein A 14 FT #SUB 4 372 MLZ F 235 337 TYR E Protein A 3 FT #SUB 5 373 LYS F 233 335 TYR E Protein B 3 FT #SUB 5 373 LYS F 234 336 GLY E Protein S 1 FT #SUB 6 374 GLY F 215 317 LYS E Protein B 1 FT #HET 4 372 MLZ F 2 2501 SAH E S 2 FT DISORDER 7 10 CC SEQUENCE 6 AA (ATOM); CC LKSXKG CC !---- CC ALIGNMENT OF SEQRES AND ATOMRES CC SEQRES LKSXKGQSTY CC ATOM LKSXKG---- CC ****** SQ SEQUENCE 10 AA; MW; CN; LKSXKGQSTY //