1 YL3 ({[6-(4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}methyl)phosphonic acid 1.000 2 1MV ({[6-(4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}methanediyl)bis(phosphonic acid) 0.846 3 KF7 [(1s)-1-{[6-(4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}-2-phenylethyl]phosphonic acid 0.759 4 KFA [(1r)-1-{[6-(4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}-2-phenylethyl]phosphonic acid 0.759 5 M2V [(1r)-1-{[6-(3-chloro-4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}-2-phenylethyl]phosphonic acid 0.733 6 M2Y [(1s)-1-{[6-(3-chloro-4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}-2-phenylethyl]phosphonic acid 0.733 7 YL5 [(1r)-2-(3-fluorophenyl)-1-{[6-(4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}ethyl]phosphonic acid 0.733 8 YL2 ({[6-(4-cyclopropylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}methanediyl)bis(phosphonic acid) 0.724 9 YF7 [(1s)-1-{[6-(3-chloro-4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}-2-(3-fluorophenyl)ethyl]phosphonic acid 0.710 10 YL4 [(R)-(2,3-dihydro-1-benzofuran-5-yl){[6-(4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}methyl]phosphonic acid 0.710 11 YL6 [(1r)-1-{[6-(3-chloro-4-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino}-2-(3-fluorophenyl)ethyl]phosphonic acid 0.710