1 W19 4-{[4-(1-benzothiophen-4-yloxy)-3-chlorophenyl]amino}-N-(2-hydroxyethyl)-8,9-dihydro-7h-pyrimido[4,5-B]azepine-6-carboxamide 1.000 2 W32 4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-N-[2-(methylsulfonyl)ethyl]-8,9-dihydro-7h-pyrimido[4,5-B]azepine-6-carboxamide 0.721