1 TG3 Ethyl (4r)-4-[[(2s)-4-methyl-2-[[(2s,3r)-3-[(2-methylpropan-2-yl)oxy]-2-(phenylmethoxycarbonylamino)butanoyl]amino]pentanoyl]amino]-5-[(3s)-2-oxidanylidenepyrrolidin-3-yl]pentanoate 1.000 2 ZU5 N-[(benzyloxy)carbonyl]-O-tert-butyl-L-threonyl-N-[(1r)-4-cyclopropyl-4-oxo-1-{[(3s)-2-oxopyrrolidin-3-yl]methyl}butyl]-L-leucinamide 0.875 3 VHP N-[(benzyloxy)carbonyl]-O-tert-butyl-L-threonyl-N-{(2s)-1-hydroxy-3-[(3s)-2-oxopyrrolidin-3-yl]propan-2-yl}-L-leucinamide 0.848 4 7VW N-[(benzyloxy)carbonyl]-O-tert-butyl-L-threonyl-N-{(2s)-1-hydroxy-3-[(3s)-2-oxopyrrolidin-3-yl]propan-2-yl}-4-methyl-L-leucinamide 0.830 5 7YW O-tert-butyl-N-{[(3-chlorophenyl)methoxy]carbonyl}-L-threonyl-N-{(2s)-1-hydroxy-3-[(3s)-2-oxopyrrolidin-3-yl]propan-2-yl}-L-leucinamide 0.830 6 G85 N-[(benzyloxy)carbonyl]-O-tert-butyl-L-seryl-N-{(2r)-5-ethoxy-5-oxo-1-[(3s)-2-oxopyrrolidin-3-yl]pentan-2-yl}-L-phenylalaninamide 0.804 7 7VB N-[(benzyloxy)carbonyl]-L-valyl-N-{(2s)-1-hydroxy-3-[(3s)-2-oxopyrrolidin-3-yl]propan-2-yl}-4-methylidene-L-norvalinamide 0.723 8 VHV N-[(benzyloxy)carbonyl]-L-valyl-N-{(2s)-1-hydroxy-3-[(3s)-2-oxopyrrolidin-3-yl]propan-2-yl}-L-leucinamide 0.723 9 VJA N-[(benzyloxy)carbonyl]-L-valyl-N-{(2r)-1-hydroxy-3-[(3s)-2-oxopyrrolidin-3-yl]propan-2-yl}-L-leucinamide 0.723 10 7V2 N-[(benzyloxy)carbonyl]-L-valyl-N-{(2s)-1-hydroxy-3-[(3s)-2-oxopyrrolidin-3-yl]propan-2-yl}-4-methyl-L-leucinamide 0.708