1 T2R (1s,3ar,5s,6r,7as)-octahydro-1,6-epoxy-2-benzofuran-5-yl {(2s,3r)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]-1-phenylbutan-2-yl}carbamate 1.000 2 NJY (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl {(2s,3r)-1-(3-fluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.860 3 NKA (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl {(2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.860 4 C7U (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.854 5 MJD (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl {(2s,3r)-1-(3,5-difluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzoxazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.843 6 QK1 (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl {(2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzothiazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.840 7 QJY (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl {(2s,3r)-1-(3,5-difluorophenyl)-3-hydroxy-4-[(2-methylpropyl)({2-[(propan-2-yl)amino]-1,3-benzothiazol-6-yl}sulfonyl)amino]butan-2-yl}carbamate 0.824 8 T1R (1r,3as,5r,6s,7ar)-octahydro-1,6-epoxy-2-benzofuran-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.812 9 065 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(2s,3r)-3-hydroxy-4-(N-isobutylbenzo[D][1,3]dioxole-5-sulfonamido)-1-phenylbutan-2-ylcarbamate 0.792 10 XUY (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(1,3-benzothiazol-6-yl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.792 11 QHA (3r,3as,4r,6ar)-4-[(2-fluoroprop-2-en-1-yl)oxy]hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.788 12 ZLP (3r,3as,4r,6ar)-4-(2-methoxyethoxy)hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[(2z)-2-(methylimino)-2,3-dihydro-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.788 13 K19 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzothiazol-6-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.776 14 K20 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{(1,3-benzodioxol-5-ylsulfonyl)[(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.776 15 J5L (3r,3as,4r,6ar)-4-[2-(methylamino)-2-oxoethoxy]hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[(2z)-2-(methylimino)-2,3-dihydro-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.774 16 G8R (1r,3as,4s,6s,7ar)-octahydro-1,6-epoxy-2-benzofuran-4-yl [(2s,3r)-4-{[2-(cyclopropylamino)-1,3-benzothiazole-6-sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.769 17 A61 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-3-[(1,3-benzothiazol-6-ylsulfonyl)(2-ethylbutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate 0.760 18 K2E (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-3-[(1,3-benzodioxol-5-ylsulfonyl)(2-ethylbutyl)amino]-1-benzyl-2-hydroxypropyl}carbamate 0.760 19 C7W (3r,3as,4r,6ar)-4-(3,3,3-trifluoropropoxy)hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[2-(methylamino)-1,3-benzoxazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.759 20 017 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl(1s,2r)-3-[[(4-aminophenyl)sulfonyl](isobutyl)amino]-1-benzyl-2-hydroxypropylcarbamate 0.750 21 7O7 (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl {(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.736 22 C7J (3r,3as,4r,6as)-4-chlorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.735 23 DJR (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{isobutyl[(4-methoxyphenyl)sulfonyl]amino}propyl]carbamate 0.735 24 GRL (3as,5r,6ar)-hexahydro-2h-cyclopenta[B]furan-5-yl (2s,3s)-3-hydroxy-4-(4-(hydroxymethyl)-N-isobutylphenylsulfonamido)-1-phenylbutan-2-ylcarbamate 0.735 25 K13 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl][(2s)-2-methylbutyl]amino}-1-benzyl-2-hydroxypropyl]carbamate 0.735 26 NJM (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[{[4-(hydroxymethyl)phenyl]sulfonyl}(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.735 27 P3V (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3,3-dihydroxy-1-phenylbutan-2-yl]carbamate 0.735 28 GR5 (2ar,4s,4ar,7ar,7br)-octahydro-2h-1,7-dioxacyclopenta[Cd]inden-4-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.727 29 GR8 (2as,4r,4as,7as,7bs)-octahydro-2h-1,7-dioxacyclopenta[Cd]inden-4-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.727 30 G52 (3r,3as,3br,6as,7as)-octahydrodifuro[2,3-B:3',2'-D]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.725 31 JDV (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(4-fluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.722 32 JDY (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3-fluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.722 33 4UX (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.720 34 52U (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.720 35 A60 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-3-{[(4-aminophenyl)sulfonyl](2-ethylbutyl)amino}-1-benzyl-2-hydroxypropyl]carbamate 0.720 36 BVR [4-[[(2~{R},3~{S})-3-[[(3~{a}~{S},4~{R},6~{a}~{R})-2,3,3~{a},4,5,6~{a}-hexahydrofuro[2,3-B]furan-4-yl]oxycarbonylamino]-2-oxidanyl-4-phenyl-butyl]-(2-methylpropyl)sulfamoyl]phenyl]-oxidanyl-oxidanylidene-boron 0.720 37 G07 4-{[(2r,3s)-3-({[(3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yloxy]carbonyl}amino)-2-hydroxy-4-phenylbutyl](2-methylpropyl)sulfamoyl}benzoic acid 0.720 38 G08 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-carbamoylphenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.720 39 G10 (3r,3as,6as)-4,4-difluorohexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-4-{[(4-aminophenyl)sulfonyl](2-methylpropyl)amino}-3-hydroxy-1-phenylbutan-2-yl]carbamate 0.720 40 G89 (3r,3ar,5r,6ar)-3-hydroxyhexahydro-2h-cyclopenta[B]furan-5-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.720 41 K14 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl][(2s)-2-methylbutyl]amino}propyl]carbamate 0.720 42 K2A (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-2-hydroxy-3-({[4-(hydroxymethyl)phenyl]sulfonyl}[(2s)-2-methylbutyl]amino)propyl]carbamate 0.720 43 NJ4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.720 44 NJA (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.720 45 0TQ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-3-hydroxy-4-[({(3z)-3-[1-(methylamino)ethylidene]-2-oxo-2,3-dihydro-1h-indol-5-yl}sulfonyl)(2-methylpropyl)amino]-1-phenylbutan-2-yl}carbamate 0.717 46 G55 (5r)-1,3-dioxepan-5-yl [(1s,2r)-1-benzyl-2-hydroxy-3-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}propyl]carbamate 0.714 47 G79 (3ar,3br,4s,7ar,8as)-decahydrofuro[2,3-B][1]benzofuran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.712 48 7OA (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-4-[{[2-(cyclopropylamino)-1,3-benzothiazol-6-yl]sulfonyl}(2-methylpropyl)amino]-1-(3,5-difluorophenyl)-3-hydroxybutan-2-yl]carbamate 0.709 49 4UY (3r,3as,4r,6ar)-4-(methylamino)hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.706 50 52W (3r,3as,4s,7as)-3-hydroxyhexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.706 51 8FM (3s,3ar,5r,7as,8s)-hexahydro-4h-3,5-methanofuro[2,3-B]pyran-8-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.706 52 B4R {4-[{(2r,3s)-3-[({[(3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl]oxy}carbonyl)amino]-2-hydroxy-4-phenylbutyl}(2-methylpropyl)sulfamoyl]phenyl}boronic acid 0.706 53 F53 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(1s,2r)-1-benzyl-3-[(2-ethylbutyl){[4-(hydroxymethyl)phenyl]sulfonyl}amino]-2-hydroxypropyl}carbamate 0.706 54 FQ4 (3as,4s,7ar)-hexahydro-4h-furo[2,3-B]pyran-4-yl [(2s,3r)-1-(4-fluorophenyl)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}butan-2-yl]carbamate 0.706 55 G04 (3r,3as,4r,6ar)-4-methoxyhexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(4-methoxyphenyl)sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.706 56 K2D (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(1s,2r)-1-benzyl-3-{(2-ethylbutyl)[(4-methoxyphenyl)sulfonyl]amino}-2-hydroxypropyl]carbamate 0.706 57 NE7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1r)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.706 58 NEJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{({4-[(1s)-1-hydroxyethyl]phenyl}sulfonyl)[(2s)-2-methylbutyl]amino}-1-phenylbutan-2-yl]carbamate 0.706 59 NF7 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1r)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.706 60 NG4 (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl {(2s,3r)-4-[({4-[(1s)-1,2-dihydroxyethyl]phenyl}sulfonyl)(2-methylpropyl)amino]-3-hydroxy-1-phenylbutan-2-yl}carbamate 0.706 61 YUJ (3r,3as,6ar)-hexahydrofuro[2,3-B]furan-3-yl [(2s,3r)-3-hydroxy-4-{[(1s)-1-hydroxy-2,3-dihydro-1h-indene-5-sulfonyl](2-methylpropyl)amino}-1-phenylbutan-2-yl]carbamate 0.706