1 SR2 (2e)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4-(dimethylamino)but-2-enamide 1.000 2 DJK N-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamide 0.852 3 YUN N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide 0.852 4 RBS N-(4-phenylamino-quinazolin-6-yl)-acrylamide 0.815 5 0WM (2e)-N-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)but-2-enamide 0.743 6 0WN N-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)butanamide 0.743 7 93J (2e)-N-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide 0.714