1 R83 N-{2,4-dimethoxy-5-[(2-piperidin-1-ylbenzyl)sulfamoyl]phenyl}acetamide 1.000 2 R84 4-{[1-(2-{[({5-[(3-carboxypropanoyl)amino]-2,4-dimethoxyphenyl}sulfonyl)amino]methyl}phenyl)piperidin-4-yl]methoxy}-4-oxobutanoic acid 0.705