1 R4J [(2r)-5-chloro-7-{2-[(2s)-1-chloro-2,3-dihydroxypropan-2-yl]thieno[3,2-B]pyridin-7-yl}-2,3-dihydro-1-benzofuran-2-yl](piperazin-1-yl)methanone 1.000 2 R41 [(2r)-7-(2-aminopyridin-4-yl)-5-chloro-2,3-dihydro-1-benzofuran-2-yl](piperazin-1-yl)methanone 0.706 3 R44 1-({7-[(2r)-5-chloro-2-(piperazine-1-carbonyl)-2,3-dihydro-1-benzofuran-7-yl]thieno[3,2-B]pyridin-2-yl}methyl)-1h-pyrrole-2,5-dione 0.700