1 OWG 3-{5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl}-1-[(1s)-6,7-dimethoxy-1-(4-methoxyphenyl)-3,4-dihydrophthalazin-2(1h)-yl]propan-1-one 1.000 2 34R (2e)-3-{5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl}-1-[(1r)-1-phenylphthalazin-2(1h)-yl]prop-2-en-1-one 0.867 3 34S (2e)-3-{5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl}-1-[(1s)-1-phenylphthalazin-2(1h)-yl]prop-2-en-1-one 0.867 4 OWM (2e)-1-[(1r)-1-cyclopropyl-6,7-dimethoxyphthalazin-2(1h)-yl]-3-{5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl}prop-2-en-1-one 0.848 5 OWS (2e)-3-{5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl}-1-[(1s)-1-(4-methylphenyl)phthalazin-2(1h)-yl]prop-2-en-1-one 0.848 6 R0Y (2e)-1-[(1s)-1-cyclopropyl-6,7-dimethoxy-3,4-dihydrophthalazin-2(1h)-yl]-3-{5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl}prop-2-en-1-one 0.848 7 OWJ (2e)-3-{5-[(2,4-diaminopyrimidin-5-yl)methyl]-2,3-dimethoxyphenyl}-1-[(1s)-1-(3,5-dimethylphenyl)phthalazin-2(1h)-yl]prop-2-en-1-one 0.830