1 MKZ 1-[4-[6-chloranyl-7-(5-methyl-1~{H}-indazol-4-yl)quinazolin-4-yl]piperazin-1-yl]propan-1-one 1.000 2 8YD 1-{4-[6-chloro-8-fluoro-7-(5-methyl-1h-indazol-4-yl)quinazolin-4-yl]piperazin-1-yl}propan-1-one 0.969 3 8YA 3-amino-1-{4-[6-chloro-8-fluoro-7-(5-methyl-1h-indazol-4-yl)quinazolin-4-yl]piperazin-1-yl}propan-1-one 0.939 4 V52 1-[(7s)-11-chloro-12-(5-methyl-1h-indazol-4-yl)-9-oxa-2,5,15,17-tetrazatetracyclo[8.7.1.02,7.014,18]octadeca-1(17),10,12,14(18),15-pentaen-5-yl]prop-2-en-1-one 0.939 5 VLE 1-[(6as)-3-chloro-2-(5-methyl-1h-indazol-4-yl)-5,6,6a,7,9,10-hexahydro-8h-pyrazino[1',2':5,6][1,5]oxazocino[4,3,2-de]quinazolin-8-yl]-2-propen-1-one 0.912 6 MKW 1-[(7r)-16-chloro-15-(5-methyl-1h-indazol-4-yl)-9-oxa-2,5,12-triazatetracyclo[8.8.0.02,7.013,18]octadeca-1(10),11,13,15,17-pentaen-5-yl]prop-2-en-1-one 0.882 7 PQI 1-[(4~{a}~{S})-7-chloranyl-8-(5-methyl-2~{H}-indazol-4-yl)-1,2,4,4~{a},5,11-hexahydropyrazino[2,1-C][1,4]benzoxazepin-3-yl]propan-1-one 0.848 8 8ZG 1-{4-[6-chloro-7-(2-fluorophenyl)quinazolin-4-yl]piperazin-1-yl}propan-1-one 0.844 9 94C 1-[4-[6-chloranyl-8-fluoranyl-7-(2-fluorophenyl)quinazolin-4-yl]piperazin-1-yl]propan-1-one 0.818 10 94F 1-[4-[6-chloranyl-8-fluoranyl-7-[2-(trifluoromethyl)phenyl]quinazolin-4-yl]piperazin-1-yl]propan-1-one 0.800 11 91S (S)-1-{4-[6-chloro-8-fluoro-7-(2-fluoro-6-hydroxyphenyl)quinazolin-4-yl] piperazin-1-yl}propan-1-one 0.794 12 V4T 1-[(4r,7s)-12-chloro-14-fluoro-13-(2-fluoro-6-hydroxyphenyl)-4-methyl-10-oxa-2,5,16,18-tetrazatetracyclo[9.7.1.0^(2,7).0^(15,19)]nonadeca-1(18),11,13,15(19),16-pentaen-5-en-1-one-yl]prop-2 0.711