1 JLE (2~{R})-2-[[6-ethyl-5-(1~{H}-indol-4-yl)thieno[2,3-D]pyrimidin-4-yl]amino]-3-phenyl-propanoic acid 1.000 2 JLK (2~{R})-2-[[6-ethyl-5-(2-methylphenyl)thieno[2,3-D]pyrimidin-4-yl]amino]-3-phenyl-propanoic acid 0.879 3 U6Q (2~{R})-2-[[5-(3-chloranyl-2-methyl-phenyl)-6-ethyl-thieno[2,3-D]pyrimidin-4-yl]amino]-3-phenyl-propanoic acid 0.853 4 U6N (2~{R})-2-[[7-but-2-ynyl-5-(3-chloranyl-2-methyl-phenyl)-6-ethyl-pyrrolo[2,3-D]pyrimidin-4-yl]amino]-3-phenyl-propanoic acid 0.718